Company Name: |
Shanghai Hongye Biotechnology Co. Ltd
|
Tel: |
400-9205774 |
Email: |
sales@glpbio.cn |
Products Intro: |
Product Name:MRS 5698 CAS:1377273-00-1 Purity:>98% Package:1mg;10mg;50mg;100mg;
|
Company Name: |
BOC Sciences
|
Tel: |
|
Email: |
info@bocsci.com |
Products Intro: |
Product Name:MRS 5698 CAS:1377273-00-1 Purity:≥96% by HPLC Remarks:MRS 5698 is a high affinity and selective A3 adenosine receptor agonist (Ki ~ 3 nM), with >1000-fold selectivity over A1 and A2A adenosine receptors. It is becoming an important pharmacological tool f
|
|
| (1S,2R,3S,4R,5S)-4-[6-[[(3-Chlorophenyl)methyl]amino]-2-[2-(3,4-difluorophenyl)ethynyl]-9H-purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide Basic information |
Product Name: | (1S,2R,3S,4R,5S)-4-[6-[[(3-Chlorophenyl)methyl]amino]-2-[2-(3,4-difluorophenyl)ethynyl]-9H-purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide | Synonyms: | (1S,2R,3S,4R,5S)-4-[6-[[(3-Chlorophenyl)methyl]amino]-2-[2-(3,4-difluorophenyl)ethynyl]-9H-purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide;MRS 5698;Bicyclo[3.1.0]hexane-1-carboxamide, 4-[6-[[(3-chlorophenyl)methyl]amino]-2-[2-(3,4-difluorophenyl)ethynyl]-9H-purin-9-yl]-2,3-dihydroxy-N-methyl-, (1S,2R,3S,4R,5S)- | CAS: | 1377273-00-1 | MF: | C28H23ClF2N6O3 | MW: | 564.97 | EINECS: | | Product Categories: | | Mol File: | 1377273-00-1.mol | |
| (1S,2R,3S,4R,5S)-4-[6-[[(3-Chlorophenyl)methyl]amino]-2-[2-(3,4-difluorophenyl)ethynyl]-9H-purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide Chemical Properties |
density | 1.58±0.1 g/cm3(Predicted) | storage temp. | Store at -20°C | solubility | Soluble in DMSO | pka | 13.31±0.70(Predicted) |
| (1S,2R,3S,4R,5S)-4-[6-[[(3-Chlorophenyl)methyl]amino]-2-[2-(3,4-difluorophenyl)ethynyl]-9H-purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide Usage And Synthesis |
Uses | MRS 5698, is a selective A3 adenosine receptor agonist, that reverses mechanoallodynia in several neuropathic pain models in vivo, and it’s orally bioavailable. | storage | Store at -20°C |
| (1S,2R,3S,4R,5S)-4-[6-[[(3-Chlorophenyl)methyl]amino]-2-[2-(3,4-difluorophenyl)ethynyl]-9H-purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide Preparation Products And Raw materials |
|