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Product Name:Benzo[3,4]cyclohept[1,2-d]imidazole, 1,4,5,6-tetrahydro-9-methyl-2-(3-pyridinyl)- CAS:447405-11-0 Purity:1020RMB/1mg Package:>98%
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BOC Sciences
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Product Name:FR252384 CAS:447405-11-0 Remarks:FR252384 is novel potent antagonists of human neuropeptide Y-Y5 receptor (IC50= 2.3 nM).
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| Benzo[3,4]cyclohept[1,2-d]imidazole, 1,4,5,6-tetrahydro-9-methyl-2-(3-pyridinyl)- Basic information |
Product Name: | Benzo[3,4]cyclohept[1,2-d]imidazole, 1,4,5,6-tetrahydro-9-methyl-2-(3-pyridinyl)- | Synonyms: | Benzo[3,4]cyclohept[1,2-d]imidazole, 1,4,5,6-tetrahydro-9-methyl-2-(3-pyridinyl)-;FR252384 | CAS: | 447405-11-0 | MF: | C18H17N3 | MW: | 275.35 | EINECS: | | Product Categories: | | Mol File: | 447405-11-0.mol | |
| Benzo[3,4]cyclohept[1,2-d]imidazole, 1,4,5,6-tetrahydro-9-methyl-2-(3-pyridinyl)- Chemical Properties |
Boiling point | 566.9±38.0 °C(Predicted) | density | 1.196±0.06 g/cm3(Predicted) | storage temp. | Store at -20°C | solubility | Soluble in DMSO | pka | 12.46±0.20(Predicted) |
| Benzo[3,4]cyclohept[1,2-d]imidazole, 1,4,5,6-tetrahydro-9-methyl-2-(3-pyridinyl)- Usage And Synthesis |
Description | FR252384 is a neuropeptide Y-Y5 receptor antagonist, with an IC50 of 2.3 nM. FR252384 is orally absorbable and permeable to brain[1]. | References | [1]. Satoh Y, et al. Novel potent antagonists of human neuropeptide Y-Y5 receptor. Part 4: tetrahydrodiazabenzazulene derivatives. Bioorg Med Chem Lett. 2002 Apr 8;12(7):1009-11. |
| Benzo[3,4]cyclohept[1,2-d]imidazole, 1,4,5,6-tetrahydro-9-methyl-2-(3-pyridinyl)- Preparation Products And Raw materials |
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