Urotensin II (114-124), human TFA
中文名称 | Urotensin II (114-124), human TFA |
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中文同义词 | |
英文名称 | Urotensin II (114-124), human TFA |
英文同义词 | Urotensin II (114-124), human TFA |
CAS号 | |
分子式 | C??H??F?N??O??S? |
分子量 | 0 |
EINECS号 | |
相关类别 | |
Mol文件 | Mol File |
结构式 |
Urotensin II (114-124), human TFA 性质
形态 | 固体 |
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颜色 | 白色至米白色 |
GPR14
Human Urotensin II (U-II) binds to recombinant human GPR14 with high affinity, and the binding is functionally coupled to calcium mobilization. Human Urotensin II induces concentration-dependent increases in intracellular calcium in a HEK-293 cell line expressing human GPR14 (EC 50 =0:62±0.17 nM, n=6).
Human Urotensin II (U-II) markedly increases total peripheral resistance in anaesthetized non-human primates, a response associated with profound cardiac contractile dysfunction.