| Company Name: |
MedChemexpress LLC
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| Tel: |
021-58955995 |
| Email: |
sales@medchemexpress.cn |
| Products Intro: |
Product Name:Pemafibrate (racemate)
CAS:848258-31-1
Purity:>98% Package:900RMB/1mg
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| Company Name: |
Musechem
|
| Tel: |
+1-800-259-7612 |
| Email: |
info@musechem.com |
| Products Intro: |
Product Name:Pemafibrate racemate
CAS:848258-31-1
Purity:>98% HPLC Package:10mg;100mg;1g Remarks:Reagent Grade
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| | Pemafibrate (racemate) Basic information |
| Product Name: | Pemafibrate (racemate) | | Synonyms: | Pemafibrate (racemate);Butanoic acid, 2-[3-[[2-benzoxazolyl[3-(4-methoxyphenoxy)propyl]amino]methyl]phenoxy]-;K13675 (racemate);2-[3-[[1,3-benzoxazol-2-yl-[3-(4-methoxyphenoxy)propyl]amino]methyl]phenoxy]butanoic acid;Pemafibrate Impurity | | CAS: | 848258-31-1 | | MF: | C28H30N2O6 | | MW: | 490.55 | | EINECS: | | | Product Categories: | | | Mol File: | 848258-31-1.mol |  |
| | Pemafibrate (racemate) Chemical Properties |
| storage temp. | Store at -20°C | | solubility | Soluble in DMSO |
| | Pemafibrate (racemate) Usage And Synthesis |
| Description | Pemafibrate racemate is the racemate of pemafibrate, and activates PPARα activity, with EC50s of 1 nM, >10 μM and 1.7 μM for h-PPARα, h-PPARγ and h-PPARδ, respectively.
h-PPARα|1 nM (EC50)|h-PPARδ|1.7 μM (EC50)
Pemafibrate racemate activates PPARα activity, with EC50s of 1 nM, >10 μM and 1.7 μM for h-PPARα, h-PPARγ and h-PPARδ, respectively[1]. | | References | [1]. Yamazaki Y, et al. Design and synthesis of highly potent and selective human peroxisome proliferator-activated receptor alpha agonists. Bioorg Med Chem Lett. 2007 Aug 15;17(16):4689-93. Epub2007 May 24. |
| | Pemafibrate (racemate) Preparation Products And Raw materials |
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