| Company Name: |
TargetMol Chemicals Inc.
|
| Tel: |
15002134094 |
| Email: |
marketing@targetmol.cn |
| Products Intro: |
Product Name:Leucettinib-92
CAS:2732859-57-1
Package:5mg;50mg
|
| Company Name: |
Adipogen Life Sciences
|
| Tel: |
41-6192660-40 |
| Email: |
info@adipogen.com |
| Products Intro: |
Product Name:Leucettinib-92
|
Leucettinib-92 manufacturers
- Leucettinib-92
-
- $0.00 / 5mg
-
2024-10-24
- CAS:2732859-57-1
- Min. Order:
- Purity:
- Supply Ability: 10g
|
| | Leucettinib-92 Basic information |
| | Leucettinib-92 Chemical Properties |
| | Leucettinib-92 Usage And Synthesis |
| Uses | Leucettinib-92 (compound 92) is an inhibitor of DYRK/CLK kinase, The IC50s are 147 nM (CLK1), 39 nM (CLK2), 5.2 nM (CLK4), 0.8 μM (CLK3), 124 nM (DYRK1A), 204 nM (DYRK1B), 0.16 μM (DYRK2), respectively. 1.0 μM (DYRK3), 0.52 μM (DYRK4), 2.78 μM (GSK3)[1]. | | References | [1] Deau E, et al. Leucettinibs, a Class of DYRK/CLK Kinase Inhibitors Inspired by the Marine Sponge Natural Product Leucettamine B. J Med Chem. 2023 Aug 10;66(15):10694-10714. DOI:10.1021/acs.jmedchem.3c00884 |
| | Leucettinib-92 Preparation Products And Raw materials |
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