| Crotonyl fentanyl Basic information |
Product Name: | Crotonyl fentanyl | Synonyms: | Crotonyl fentanyl;Crotonyl fentanyl (CRM);2-Butenamide, N-phenyl-N-[1-(2-phenylethyl)-4-piperidinyl]-, (2E)- | CAS: | 760930-59-4 | MF: | C23H28N2O | MW: | 348.48 | EINECS: | | Product Categories: | | Mol File: | 760930-59-4.mol | ![Crotonyl fentanyl Structure](CAS/20181012/GIF/760930-59-4.gif) |
| Crotonyl fentanyl Chemical Properties |
solubility | DMF: 30 mg/ml; DMSO: 20 mg/ml; Ethanol: 30 mg/ml; PBS (pH 7.2): 10 mg/ml | form | A neat solid |
DEA Controlled Substances | CSCN: 9844 CSA SCH: Schedule I NARC: Yes |
| Crotonyl fentanyl Usage And Synthesis |
Description | Crotonyl fentanyl is an analytical reference material categorized as an opioid.1,2,3 Crotonyl fentanyl induces generalized responses in mice trained to discriminate oxycodone from saline.4 Crotonyl fentanyl is regulated as a Schedule I compound in the United States. This product is intended for research and forensic applications. | Uses | Crotonyl Fentanyl is an analog of Fentanyl (F274990), which is a controlled substanced used as analgesic. | References | 1. Eshleman, A.J., Nagarajan, S., Wolfrum, K.M., et al. Affinity, potency, efficacy, selectivity, and molecular modeling of substituted fentanyls at opioid receptors Biochem. Pharmacol. 182,114293(2020). 2. Vasudevan, L., Vandeputte, M.M., Deventer, M., et al. Assessment of structure-activity relationships and biased agonism at the mu opioid receptor of novel synthetic opioids using a novel, stable bio-assay platform Biochem. Pharmacol. 177,113910(2020). 3. Varshneya, N.B., Walentiny, D.M., Moisa, L.T., et al. Opioid-like antinociceptive and locomotor effects of emerging fentanyl-related substances Neuropharmacology 151,171-179(2019). 4. Walentiny, D.M., Moisa, L.T., and Beardsley, P.M. Oxycodone-like discriminative stimulus effects of fentanyl-related emerging drugs of abuse in mice Neuropharmacology 150,210-216(2019). |
| Crotonyl fentanyl Preparation Products And Raw materials |
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