Autocamtide-2-related inhibitory peptide TFA
中文名称 | Autocamtide-2-related inhibitory peptide TFA |
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中文同义词 | |
英文名称 | Autocamtide-2-related inhibitory peptide TFA |
英文同义词 | Autocamtide-2-related inhibitory peptide TFA |
CAS号 | |
分子式 | C??H???N??O??F? |
分子量 | 0 |
EINECS号 | |
相关类别 | |
Mol文件 | Mol File |
结构式 |
Autocamtide-2-related inhibitory peptide TFA 性质
形态 | 固体 |
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颜色 | 白色至米白色 |
Autocamtide-2-related inhibitory peptide (TFA) 是高度特异性的、CaMKII 的有效抑制剂,其 IC50 值为 40 nM。
IC50: 40 nM (CaMKII).
It is found that Autocamtide-2-related inhibitory peptide (TFA) is a potent inhibitor of CaM-kinase II with an IC 50 of 40 nM, which is active in the presence or absence of Ca 2+ /calmodulin. It is 50 and 500 times more potent than CaMK-(281-302Ala286) and KN-93, respectively, under the assay condition used.