Product Details
Product Name:
NEO2734 |
CAS No.:
2081072-29-7 |
Purity:
98.80% |
Supply Ability:
10g |
Release date:
2024/11/04 |
Product Introduction
Bioactivity
名称 | NEO2734 |
描述 | NEO2734 (EP31670) is an orally active, selective inhibitor of p300/CBP and BET bromodomains, with an IC50 of less than 30 nM for both targets. |
体外活性 | NEO2734, a novel dual inhibitor of BET and CBP/p300, is active in both hotspot mutant (F133V) and non-hotspot mutant (Q165P) PCa cells in vitro and in vivo[1]. |
存储条件 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
溶解度 | DMSO : 27.5 mg/mL (63.15 mM)
|
关键字 | NEO-2734 | PER-403 | SPOP | CBP | MYC | HAT | Epigenetic Reader Domain | NEO 2734 | TC-797 | Histone Acetyltransferase | p300 | HATs | inhibit | Inhibitor | EP 31670 | EP-31670 | NEO2734 |
相关产品 | ABBV-744 | CeMMEC1 | 3-methyl-1,2,3,4-tetrahydroquinazolin-2-one | (+)-JQ-1 | J-147 | Anacardic Acid | Acetaminophen | Curcumin | dBET6 | Piflufolastat | Naphthol AS-E | Bisdemethoxycurcumin |
相关库 | 组蛋白修饰化合物库 | 表型筛选靶点鉴定库 | 经典已知活性库 | 表观遗传库 | 抑制剂库 | PPI抑制剂库 | 口服活性化合物库 | 已知活性化合物库 | 抗癌化合物库 | 抗癌活性化合物库 |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
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Recommended supplier
Product name |
Price |
|
Suppliers |
Update time |
|
$/ |
|
Anhui Ruihan Technology Co., Ltd
|
2023-08-21 |