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  •       科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。
英文名称 中文名称 CAS号 操作
ethyl 3-oxo-8-azabicyclo[3.2.1]octane-8-carboxylate 3-氧代去甲托烷-8-羧酸乙酯 32499-64-2 详细
(1R,4S)-7,7-dimethyl-2-oxo-norbornan-1-yl]methanesulfonic acid 左旋樟脑磺酸 35963-20-3 详细
tert-butyl 3-aminobicyclo[1.1.1]pentane-1-carboxylate 叔-丁基 3-氨基二环[1.1.1]戊烷-1-甲酸基酯 1935523-60-6 详细
8-thia-3-azabicyclo[3.2.1]octane 280-25-1 详细
(1R)-2-azabicyclo[2.2.1]heptane-4-carboxylic acid;hydrochloride (1R)-2-氮杂双环[2.2.1]庚烷-4-羧酸盐酸盐 1212489-75-2 详细
1-{bicyclo[2.2.1]heptan-2-yl}ethan-1-amine 1-二环[2.2.1]庚-2-基乙胺 24520-60-3 详细
methyl (2S)-2-(benzyloxycarbonylamino)-3-(1-bicyclo[1.1.1]pentanyl)propanoate 2940861-58-3 详细
dimethyl 3-oxabicyclo[3.1.1]heptane-1,5-dicarboxylate 2920404-85-7 详细
3,7-dipropyl-3,7-diazabicyclo[3.3.1]nonane 3,7-二丙基-3,7-二氮杂二环[3.3.1]壬烷 909037-18-9 详细
tert-butyl 6-oxa-3-azabicyclo[3.1.1]heptane-3-carboxylate 6-氧杂-3-氮杂双环[3.1.1]庚烷-3-羧酸叔丁酯 1305208-01-8 详细
1-(1-adamantyl)ethanamine;hydrochloride 盐酸金刚乙胺 1501-84-4 详细
ethyl 1-azabicyclo[2.2.1]heptane-4-carboxylate 1-氮杂双环[2.2.1]庚烷-4-羧酸乙酯 119102-24-8 详细
7-oxabicyclo[2.2.1]heptan-2-one 58564-88-8 详细
5-hydroxybicyclo[3.1.1]heptane-1-carboxylic acid 2091096-37-4 详细
bicyclo[3.1.1]heptane-1-carboxylic acid 双环[3.1.1]庚烷-1-羧酸 91239-72-4 详细
4-{[(tert-butoxy)carbonyl]amino}-2-oxabicyclo[2.2.2]octane-1-carboxylic acid 4-((叔丁氧基羰基)氨基)-2-氧杂二环[2.2.2]辛烷-1-羧酸 2010218-26-3 详细
5-bromobicyclo[3.1.1]heptane-1-carboxylic acid 168974-64-9 详细
tert-butyl 1-(hydroxymethyl)-2-azabicyclo[2.2.1]heptane-2-carboxylate 1780679-52-8 详细
6-tert-butoxycarbonyl-6-azabicyclo[3.1.1]heptane-1-carboxylic acid 6-叔丁氧基羰基-6-氮杂双环[3.1.1]庚烷-1-羧酸 2680539-11-9 详细
3-(tert-butoxycarbonylamino)-2,2-difluoro-bicyclo[1.1.1]pentane-1-carboxylic acid 2408970-21-6 详细
1-(difluoromethyl)-2-oxabicyclo[2.2.2]octan-4-amine;hydrochloride 2170372-49-1 详细
7-oxabicyclo[2.2.1]heptan-1-ylmethanamine;hydrochloride 2624140-49-2 详细
2-(benzyloxycarbonylamino)-3-(1-bicyclo[1.1.1]pentanyl)propanoic acid 2940934-29-0 详细
5-aminonorpinan-1-ol;hydrochloride 2940947-90-8 详细
3-oxabicyclo[3.1.1]heptan-1-ylmethyl 4-methylbenzenesulfonate 2955561-33-6 详细
methyl 4-{[(benzyloxy)carbonyl]amino}bicyclo[2.2.2]octane-1-carboxylate 甲基 4-{[(苄氧基)羰基]氨基}二环[2.2.2]辛烷-1-甲酸基酯 862501-91-5 详细
bicyclo[3.2.1]octane-3-carboxylic acid bicyclo[3.2.1]octane-3-carboxylic acid 6221-65-4 详细
tert-butyl exo-3-hydroxy-9-azabicyclo[3.3.1]nonane-9-carboxylate 叔-丁基外-3-羟基-9-氮杂二环[3.3.1]壬烷-9-甲酸基酯 934233-73-5 详细
2-azabicyclo[2.2.2]octane-4-carboxylic acid;hydrochloride 2-azabicyclo[2.2.2]octane-4-carboxylic acid hydrochloride 1394042-79-5 详细
2-[(tert-butoxy)carbonyl]-2-azabicyclo[2.2.2]octane-5-carboxylic acid 2-[(tert-butoxy)carbonyl]-2-azabicyclo[2.2.2]octane-5-carboxylic acid 1890098-49-3 详细
tert-butyl N-(5-aminonorpinan-1-yl)carbamate (5-氨基双环[3.1.1]庚-1-基)氨基甲酸叔丁酯 1049607-15-9 详细
(4-amino-2-oxabicyclo[2.1.1]hexan-1-yl)methanol {4-氨基-2-氧杂双环[2.1.1]己-1-基}甲醇 2170372-31-1 详细
methyl 3-oxabicyclo[3.1.1]heptane-1-carboxylate 2940950-46-7 详细
tert-butyl endo-3-hydroxy-6-azabicyclo[3.1.1]heptane-6-carboxylate ENDO-3-羟基-6-氮杂双环[3.1.1]庚烷-6-羧酸叔丁酯 2982738-99-6 详细
(1S,4S)-2-methyl-2,5-diazabicyclo[2.2.1]heptane dihydrobromide (1S,4S)-2-甲基-2,5-二氮杂二环[2.2.1]庚二氢溴酸盐 125224-62-6 详细
tert-butyl 3-hydroxy-3-methyl-8-azabicyclo[3.2.1]octane-8-carboxylate 3-羟基-3-甲基-8-氮杂双环[3.2.1]辛烷-8-甲酸叔丁酯 870889-20-6 详细
6-azabicyclo[3.2.1]octan-3-one;hydrochloride 6-氮杂双环[3.2.1]辛-3-酮盐酸盐 1378821-66-9 详细
tert-butyl exo-3-(hydroxymethyl)-8-azabicyclo[3.2.1]octane-8-carboxylate 外-8-boc-8-氮杂二环[3.2.1]辛烷-3-甲醇 273207-58-2 详细
4-(benzyloxycarbonylamino)norbornane-1-carboxylic acid 1252672-36-8 1252672-36-8 详细
rel-(1S,3S,4S,5R)-2-tert-butoxycarbonyl-5-hydroxy-2-azabicyclo[2.2.1]heptane-3-carboxylic acid (1s,3s,4s,5r)-rel-2-boc-5-羟基-2-氮杂二环[2.2.1]庚烷-3-羧酸 1290625-54-5 详细
4-benzyl-1,4-diazabicyclo[3.2.1]octane 4-苄基-1,4-二氮杂双环螺[3.2.1]辛烷 675589-81-8 详细
4-bromobicyclo[2.2.1]heptane-1-carboxylic acid 4-溴二环[2.2.1]庚烷-1-羧酸 15448-85-8 详细
3,5-dimethyladamantane-1-carboxylic acid 3,5-二甲基金刚烷-1-羧酸 14670-94-1 详细
endo-tert-butyl 8-hydroxy-3-azabicyclo[3.2.1]octane-3-carboxylate endo-tert-butyl 8-hydroxy-3-azabicyclo[3.2.1]octane-3-carboxylate 1246947-33-0 详细
3,9-dioxa-7-azabicyclo[3.3.1]nonane hydrochloride 3,9-dioxa-7-azabicyclo[3.3.1]nonane hydrochloride 1803587-96-3 详细
1-methyl-2-oxabicyclo[2.1.1]hexane-4-carboxylic acid 1-methyl-2-oxabicyclo[2.1.1]hexane-4-carboxylic acid 2169582-80-1 详细
4-amino-2-oxabicyclo[2.1.1]hexane-1-carbonitrile hydrochloride 4-氨基-2-氧杂双环[2.1.1]己烷-1-甲腈盐酸盐 2170372-36-6 详细
3-methoxy-N-methyl-bicyclo[1.1.1]pentan-1-amine;hydrochloride (3-甲氧基-双环[1.1.1]戊-1-基)-甲胺盐酸盐 2752941-70-9 详细
methyl 4-(hydroxymethyl)cubane-1-carboxylate 4-羟甲基-立方烷-1-羧酸甲基酯 60462-19-3 详细
4-oxoadamantane-1-carboxylic acid 2-金刚烷酮-5-甲酸 56674-87-4 详细
methyl 5-(hydroxymethyl)bicyclo[3.1.1]heptane-1-carboxylate 5-(羟甲基)双环[3.1.1]庚烷-1-羧酸甲酯 2091771-31-0 详细
3-oxabicyclo[3.1.1]heptane-1-carboxylic acid 3-氧杂环[3.1.1]庚烷-1-羧酸 2490375-56-7 详细
(5-methyl-3-oxabicyclo[3.1.1]heptan-1-yl)methanol 2920401-68-7 详细
2-[(1S,4S)-2-oxa-5-azabicyclo[2.2.1]heptan-5-yl]ethanol;oxalic acid 2940861-54-9 详细
tert-butyl N-(8-azabicyclo[3.2.1]octan-3-yl)carbamate 3-叔丁氧酰基氨基脱甲托品烷 287114-25-4 详细
tert-butyl 3,7-diazabicyclo[3.3.1]nonane-3-carboxylate 7-叔丁氧羰基-3,7-二氮杂双环[3.3.1]壬烷 227940-72-9 详细
tert-butyl anti-7-amino-2-azabicyclo[2.2.1]heptane-2-carboxylate REL-(1R,4R,7R)-7-氨基-2-氮杂双环[2.2.1]庚烷-2-羧酸叔丁酯 1290626-52-6 详细
5-aminonorpinan-1-ol 5-aminobicyclo[3.1.1]heptan-1-ol 2091526-30-4 详细
4-(trifluoromethyl)bicyclo[2.2.2]octan-1-yl]methanol [4-(trifluoromethyl)bicyclo[2.2.2]octan-1-yl]methanol 94994-14-6 详细
(1R,4R)-2-oxa-5-azabicyclo[2.2.2]octane;hydrochloride (1R,4R)-2-OXA-5-AZABICYCLO[2.2.2] 辛烷,氯化氢 (1:1) 2306254-89-5 详细
8-thia-3-azabicyclo[3.2.1]octane;hydrochloride 8-硫杂-3-氮杂双环[3.2.1]辛烷盐酸盐 16074-68-3 详细
(1S,4S)-2-oxa-5-azabicyclo[2.2.2]octane;hydrochloride (1S,4S)-2-OXA-5-AZABICYCLO[2.2.2]辛烷,氯化氢(1:1) 2306249-59-0 详细
endo-N-methylnorbornan-2-amine;hydrochloride 内向-N-甲基双环[2.2.1]庚烷-2-胺盐酸盐 131274-98-1 详细
(2R)-2-(benzyloxycarbonylamino)-3-(1-bicyclo[1.1.1]pentanyl)propanoic acid 2322921-14-0 详细
methyl 4-(methoxymethyl)norbornane-1-carboxylate 2725791-10-4 详细
ethyl (1R,2S,5S)-3,8-diazabicyclo[3.2.1]octane-2-carboxylate;dihydrochloride 2940857-56-5 详细
tert-butyl N-(3-oxabicyclo[3.1.1]heptan-1-ylmethyl)carbamate 2970213-92-2 详细
4-fluoro-2-azabicyclo[2.1.1]hexane-1-carboxylic acid 4-氟-2-氮杂双环[2.1.1]己烷-1-羧酸 1196976-68-7 详细
(1R)-1-(adamantan-1-yl)ethan-1-amine hydrochloride (R)-1-(金刚烷-1-基)乙胺盐酸盐 1005341-52-5 详细
methyl 4-{[(benzyloxy)carbonyl]amino}bicyclo[2.2.1]heptane-1-carboxylate methyl 4-(((benzyloxy)carbonyl)amino)bicyclo[2.2.1]heptane-1-carboxylate 1252672-35-7 详细
tert-butyl 3,9-diazabicyclo[4.2.1]nonane-3-carboxylate 叔-丁基 3,9-二氮杂二环[4.2.1]壬烷-3-甲酸基酯 286947-16-8 详细
endo-2-tert-butoxycarbonyl-2-azabicyclo[2.1.1]hexane-5-carboxylic acid (1r,4s,5s)-rel-2-boc-2-氮杂二环[2.1.1]己烷-5-羧酸 615575-74-1 详细
endo-8-tert-butoxycarbonyl-8-azabicyclo[3.2.1]octane-3-carboxylic acid (1R,3R,5S)-rel-8-[(叔-丁氧基)羰基]-8-氮杂二环[3.2.1]辛烷-3-羧酸 1222996-05-5 详细
exo-7-(boc-amino)-3-oxa-9-aza-bicyclo[3.3.1]nonane 外-7-(boc-氨基)-3-氧杂-9-氮杂-二环[3.3.1]壬烷 1638683-57-4 详细
tert-butyl 2-oxa-3-azabicyclo[2.2.1]hept-5-ene-3-carboxylate 2-氧杂-3-氮杂双环[2.2.1]庚-5-烯-3-羧酸叔丁酯 99027-90-4 详细
7-oxabicyclo[2.2.1]heptane-1-carboxylic acid 7-氧杂双环[2.2.1]庚烷-1-羧酸 1706450-79-4 详细
tert-butyl N-{3-methylidenebicyclo[3.2.1]octan-8-yl}carbamate 叔-丁基 N-{3-甲亚基二环[3.2.1]辛烷-8-基}氨基甲酯 2168116-64-9 详细
methyl 4-bromobicyclo[2.2.1]heptane-1-carboxylate 4-溴双环[2.2.1]庚烷-1-甲酸甲酯 15448-84-7 详细
4-hydroxybicyclo[2.2.1]heptane-1-carboxylic acid 4-hydroxybicyclo[2.2.1]heptane-1-carboxylic acid 88888-30-6 详细
2-adamantylmethanamine (2-金刚烷基甲基)胺盐酸盐 42067-67-4 详细
8-tert-butoxycarbonyl-3-oxa-8-azabicyclo[3.2.1]octane-1-carboxylic acid 3-氧杂-8-氮杂双环[3.2.1]辛烷-1,8-二羧酸-8-(1,1-二甲基乙基)酯 1638651-87-2 详细
7-oxabicyclo[2.2.1]heptan-1-ylmethanol 7-氧杂双环[2.2.1]庚烷-1-甲醇 15574-03-5 详细
1-methyl-2-oxabicyclo[2.1.1]hexan-4-amine hydrochloride 1-甲基-2-氧杂双环[2.1.1]己-4-胺盐酸盐 2170372-24-2 详细
bicyclo[2.2.1]heptane-1-carboxylic acid 1-降莰烷甲酸 18720-30-4 详细
3,6-diazabicyclo[3.1.1]heptane;dihydrochloride 2725791-26-2 详细
methyl 5-amino-3-oxabicyclo[3.1.1]heptane-1-carboxylate 2920401-64-3 详细
tert-butyl exo-6-hydroxy-2-azabicyclo[2.2.1]heptane-2-carboxylate 叔-丁基外-6-羟基-2-氮杂二环[2.2.1]庚烷-2-甲酸基酯 198835-02-8 详细
tert-butyl exo-5-hydroxy-2-azabicyclo[2.2.1]heptane-2-carboxylate rel-叔-丁基 (1S,4S,5R)-5-羟基-2-氮杂二环[2.2.1]庚烷-2-甲酸基酯 198835-03-9 详细
tert-butyl 3-amino-6-azabicyclo[3.2.1]octane-6-carboxylate (1R,3S,5R)-叔-丁基 3-氨基-6-氮杂二环[3.2.1]辛烷-6-甲酸基酯 1199942-73-8 详细
methyl 5-bromobicyclo[3.1.1]heptane-1-carboxylate Bicyclo[3.1.1]heptane-1-carboxylic acid, 5-bromo-, methyl ester 91239-76-8 详细
methyl 5-hydroxybicyclo[3.1.1]heptane-1-carboxylate 5-羟基双环[3.1.1]庚烷-1-羧酸甲酯 168974-76-3 详细
bicyclo[3.1.1]heptane-1,5-dicarboxylic acid 双环[3.1.1]庚烷-1,5-二羧酸 75328-55-1 详细
1-azabicyclo[2.2.2]octane-3-carboxylic acid 1-氮杂双环[2.2.2]辛烷-3-甲酸 75208-40-1 详细
tert-butyl N-(3-methylsulfanyl-1-bicyclo[1.1.1]pentanyl)carbamate 2940937-57-3 详细
tert-butyl 7-hydroxy-9-oxa-3-azabicyclo[3.3.1]nonane-3-carboxylate 2940940-71-4 详细
adamantan-2-amine;hydrochloride 2-金刚烷胺盐酸盐 10523-68-9 详细
norbornan-1-amine;hydrochloride 二环[2.2.1]庚烷-1-胺盐酸 75934-56-4 详细
bicyclo[2.2.1]heptan-2-ol 降冰片 1632-68-4 详细
O8-tert-butyl O3-methyl endo-8-azabicyclo[3.2.1]octane-3,8-dicarboxylate 8-叔-丁基 3-甲基内-8-氮杂二环[3.2.1]辛烷-3,8-二甲酸基酯 1548548-51-1 详细
1-(iodomethyl)-7-oxabicyclo[2.2.1]heptane 1-(碘甲基)-7-氧杂双环[2.2.1]庚烷 946402-76-2 详细
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