产品属性:
产品名称
规格
CAS号
型号
HFI-142
5mg
332164-34-8
EY-Y0164175
Cas No.332164-34-8
别名 N/A
化学名 N/A
分子式 C17H16N2O4
分子量 312.32
溶解度 Soluble in DMSO
储存条件 Store at -20°C General tips For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. Shipping Condition Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request 产品描述: HFI-142 is an insulin-regulated aminopeptidase (IRAP) inhibitor with a ki of 2.01 μM[1]. ki: 2.01 μM (Insulin-regulated aminopeptidase)[1]
[1]. Albiston AL, et al. Phenylalanine-544 plays a key role in substrate and inhibitor binding by providing a hydrophobicpacking point at the active site of insulin-regulated aminopeptidase. Mol Pharmacol. 2010 Oct;78(4):600-7.
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