Product Name:GaTx2
CAS No.:194665-85-5
Synonyms:阻断剂多肽GaTx2
Catalog No.:218P217
Brand:HongTide(上海鸿肽生物)
Description:GaTx2 是一种非常高亲和力的 ClC-2 阻断剂(表观 KD ~ 50 pM)多肽,序列中含有29个氨基酸,并且含有3对二硫键,能减缓 ClC-2 活化并抑制慢门控,但不抑制开放的 ClC-2 通道。GaTx2对 ClC-2 的选择性优于其他 ClC 家族成员(ClC-0、ClC-1、ClC-3 和 ClC-4)、CFTR、GABAC、CaCC 和 KV1.2。
GaTx2 is a highly affinity ClC-2 blocker (apparent KD~50 pM) peptide with 29 amino acids in its sequence and 3 pairs of disulfide bonds. It can slow down ClC-2 activation and inhibit slow gating, but does not inhibit open ClC-2 channels. GaTx2 has better selectivity for ClC-2 than other members of the ClC family (ClC-0, ClC-1, ClC-3, and ClC-4), CFTR, GABAC, CaCC, and KV1.2.
Purity (HPLC) ≥98.0%
Single impurity≤2%
Peptide content≥75.0%
Amino Acid Composition≤±15%
Bacterial Endotoxins≤50EU/mg
Solubility:H2O/DMSO
Vacuum-packed with aluminum foil bag or transparent bag.Various weights can be packed according to your requirements.
Storage:Cool dry place( Store at -20°C, away from the light)
Remark:For Research Use Only. Not for human use.
Sequence(1-letter code) | VSCEDCPDHCSTQKARAKCDNDKCVCEPI(Disulfide bridge:Cys3-Cys19;Cys6-Cys24;Cys10-Cys26) |
Sequence(3-letter code) | H-Val-Ser-Cys-Glu-Asp-Cys-Pro-Asp-His-Cys-Ser-Thr-Gln-Lys-Ala-Arg-Ala-Lys-Cys-Asp-Asn-Asp-Lys-Cys-Val-Cys-Glu-Pro-Ile-OH(Disulfide bridge:Cys3-Cys19;Cys6-Cys24;Cys10-Cys26) |
Peptide Structure |
|
Molecular Formula | C125H199N39O47S6 |
Molecular Weight | 3192.54 |
订购联系方式:
上海鸿肽生物科技有限公司
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QQ: 3259098395
邮箱:sales1@hongtide.com
关键字: 194665-85-5;GaTx2 ;阻断剂多肽GaTx2;多肽;多肽合成;
上海鸿肽生物科技有限公司(简称:鸿肽生物)是一家以多肽以及多肽上下游产品研发、生产、销售以及技术转让为主要业 务科技公司。公司现有产品涵盖:定制多肽、目录多肽、氨基酸衍生物、小分子化合物;公司自成立以来,秉持“用质量作船, 以服务为帆,为科研服务”的企业理念,为国内外众多科研工作者提供了优质的服务及产品。