别名
2-Amino-1,1,3-tricyano-4-(3′,4′,5′-trihydroxyphenyl)butadiene
溶解性
DMSO: soluble 5 mg of Tyrphostin 51 in 0.1 ml of solvent, clear, orange to red
应用
Tyrphostin 51 has been used to study the inhibition of rat hepatic leptin 1.
生化/生理作用
Tyrphostin 51 is a small molecule inhibitor of epidermal growth factor (EGF) receptor kinase function. This molecule associates with the substrate subsite of the protein tyrosine kinase (PTK) domain,. EGFR tyrosine kinase inhibitor.
制备说明
5 mg of Tyrphostin 51 is soluble in 0.1 ml of DMSO and yields a clear, orange to red solution.
Sigma-Aldrich西格玛奥德里奇(上海)贸易有限公司
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