中文名:WYE-687,mTOR抑制剂
英文名:WYE-687
中文别名:N-[4-[4-(4-吗啉基)-1-[1-(3-吡啶甲基)-4-哌啶基]-1H-吡唑并[3,4-D]嘧啶-6-基]苯基]氨基甲酸甲酯|N-[4-[4-(4-吗啉基)-1-[1-(3-吡啶甲基)-4-哌啶基]-1H-吡唑并[3,4-D]嘧啶-6-基]苯基]氨基甲酸甲酯
英文别名:WYE-687|1062161-90-3|methyl (4-(4-morpholino-1-(1-(pyridin-3-ylmethyl)piperidin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-6-yl)phenyl)carbamate|WYE 687|methyl N-[4-[4-morpholin-4-yl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrazolo[3,4-d]pyrimidin-6-yl]phenyl]carb
纯度:≥98%
货号:W126399
包装:50mg、5mg、25mg
Cas号:1062161-90-3
存储温度:-20°C储存
产品介绍:
WYE-687是ATP竞争性mTOR选择性抑制剂,比对PI3Kα/γ的抑制性高超过100倍。A potent ATP-competitive mTOR inhibitor with an IC50 of 7 nM
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