中文名:VUF 10166,5-HT3拮抗剂
英文名:VUF 10166
中文别名:2-氯-3-(4-甲基-1-哌嗪基)喹喔啉
英文别名:155584-74-0|2-chloro-3-(4-methylpiperazin-1-yl)quinoxaline|VUF 10166|Quinoxaline, 2-chloro-3-(4-methyl-1-piperazinyl)-|CHEMBL261010|VUF10166|VUF10166;VUF-10166|2-Chloro-3-(4-methyl-1-piperazinyl)quinoxaline|SCHEMBL404203|DTXSID60640663|HMS3651F21|HMS3884N
纯度:≥99%
货号:V129763
包装:10mg、50mg、250mg
Cas号:155584-74-0
存储温度:-20°C储存
产品介绍:
VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower. VUF10166 shows low activity to 5-HT3AB receptor with Ki of 22 nM. VUF10166 may be used to can distinguish between 5-HT3A and 5-HT3AB receptors. VUF10166 has no activity to α7 nACh receptor. VUF10166 also acts as a partial agonist at 5-HT3A receptors with EC50 of 5.2 μM, which shows that VUF10166 is unlikely to bind in the receptor pore.
查看阿拉丁官网此产品相关对应页面:https://www.aladdin-e.com/zh_cn/V129763.html
上海阿拉丁生化科技股份有限公司
联系商家时请提及chemicalbook,有助于交易顺利完成!
阿拉丁客服