JAK3:0.7 nM (IC50)
JAK1:3.9 nM (IC50)
JAK2:5 nM (IC50)
Tyk2:4.8 nM (IC50)
[1]. Ito M, et al. A novel JAK inhibitor, peficitinib, demonstrates potent efficacy in a rat adjuvant-induced arthritis model. J Pharmacol Sci. 2017 Jan;133(1):25-33.
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