Product Name:YAP-TEAD-IN-1
CAS No.:1659305-79-9(TFA);1659305-78-8
Synonyms:竞争性肽类抑制剂YAP-TEAD-IN-1
Catalog No.:218P777
Brand:HongTide(上海鸿肽生物)
Description:YAP-TEAD-IN-1 TFA 是 YAP-TEAD 相互作用的有效的竞争性肽类抑制剂,其IC50值为25 nM,是由17个氨基酸组成的多肽。YAP-TEAD-IN-1 TFA 是一种 17mer 的多肽,与 YAP (50-171) (Kd=40 nM) 相比,其与 TEAD1 的结合亲和力更高 (Kd= 15 nM)。
YAP-TEAD-IN-1 TFA is an effective competitive peptide inhibitor of YAP-TEAD interaction, with an IC50 value of 25 nM. It is a peptide composed of 17 amino acids. YAP-TEAD-IN-1 TFA is a 17 mer peptide with a higher binding affinity to TEAD1 (Kd=15 nM) compared to YAP (50-171) (Kd=40 nM).
Purity (HPLC) ≥98.0%
Single impurity≤2%
Peptide content≥75.0%
Amino Acid Composition≤±15%
Bacterial Endotoxins≤50EU/mg
Solubility:H2O/DMSO
Vacuum-packed with aluminum foil bag or transparent bag.Various weights can be packed according to your requirements.
Storage:Cool dry place( Store at -20°C, away from the light)
Remark:For Research Use Only. Not for human use.
Sequence(1-letter code) | Ac-VP-Phe(3-Cl)-Hcy-LRK-Nle-PASFCKPPE-NH2(Disulfide bridge:Hcy4-Cys13) |
Sequence(3-letter code) | Ac-Val-Pro-Phe(3-Cl)-HomoCys-Leu-Arg-Lys-Nle-Pro-Ala-Ser-Phe-Cys-Lys-Pro-Pro-Glu-NH2 (Disulfide bridge:Hcy4-Cys13) |
Peptide Structure |
|
Molecular Formula | C93H144ClN23O21S2 |
Molecular Weight | 2019.86 |
订购联系方式:
上海鸿肽生物科技有限公司
手机: +86-18018095145 (同微信号)
QQ: 3259098395
邮箱:sales1@hongtide.com
关键字: 1659305-78-8;1659305-79-9(TFA);YAP-TEAD-IN-1 ;竞争性肽类抑制剂YAP-TEAD-IN-;多肽;
上海鸿肽生物科技有限公司(简称:鸿肽生物)是一家以多肽以及多肽上下游产品研发、生产、销售以及技术转让为主要业 务科技公司。公司现有产品涵盖:定制多肽、目录多肽、氨基酸衍生物、小分子化合物;公司自成立以来,秉持“用质量作船, 以服务为帆,为科研服务”的企业理念,为国内外众多科研工作者提供了优质的服务及产品。