生物活性25-Hydroxycholesterol是胆固醇的代谢产物,由巨噬细胞响应Toll样受体(TLR)激活而产生和分泌。25-Hydroxycholesterol有效且选择性抑制B细胞产生IgA,EC50约为65nM。
靶点HumanEndogenousMetabolite
体外研究Thesynthesisof25-hydroxycholesteroliscatalyzedbytheenzymecholesterol25-hydroxylase,whichusescholesterolandmolecularoxygenassubstratesandNADPHasacofactor.25-hydroxycholesterolisapotentbioactivelipidintheinnateandadaptiveimmunesystems.
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