Product Name:L-JNKI-1
CAS No.:N/A
Synonyms:胞渗透性多肽抑制剂多肽L-JNKI-1
Catalog No.:218P872
Brand:HongTide(上海鸿肽生物)
Description:L-JNKI-1是一种针对 JNK 的细胞渗透性多肽抑制剂多肽,是由31个氨基酸组成的多肽。在体内研究中,L-JNKI-1 已被证明可有效抑制 JNK 活性。 结果表明,Ang II 诱导剂量依赖性升压反应,JNK 抑制显着减弱了该反应。 还发现 10 μM L-JNKI-1 将磷酸化 c-Jun 降低 98%,磷酸化 Elk-1 降低 100%。 L-JNKI-1能够在腹腔注射后1小时内穿过血脑屏障并穿透成年小鼠和P5大鼠的神经元
L-JNKI-1 is a cell penetrating peptide inhibitor peptide targeting JNK, composed of 31 amino acids. In vivo studies have shown that L-JNKI-1 can effectively inhibit JNK activity. The results showed that Ang II induced a dose-dependent pressor response, and JNK inhibition significantly weakened this response. It was also found that 10 μ M L-JNKI-1 reduced phosphorylated c-Jun by 98% and phosphorylated Elk-1 by 100%. L-JNKI-1 can cross the blood-brain barrier and penetrate neurons in adult mice and P5 rats within 1 hour after intraperitoneal injection
Purity (HPLC) ≥98.0%
Single impurity≤2%
Peptide content≥75.0%
Amino Acid Composition≤±15%
Bacterial Endotoxins≤50EU/mg
Solubility:H2O/DMSO
Vacuum-packed with aluminum foil bag or transparent bag.Various weights can be packed according to your requirements.
Storage:Cool dry place( Store at -20°C, away from the light)
Remark:For Research Use Only. Not for human use.
Sequence(1-letter code) | DQSRPVQPFLNLTTPRKPRPPRRRQRRKKRG-NH2 |
Sequence(3-letter code) | H-Asp-Gln-Ser-Arg-Pro-Val-Gln-Pro-Phe-Leu-Asn-Leu-Thr-Thr-Pro-Arg-Lys-Pro-Arg-Pro-Pro-Arg-Arg-Arg-Gln-Arg-Arg-Lys-Lys-Arg-Gly-NH2 |
Peptide Structure |
|
Molecular Formula | C164H286N66O40 |
Molecular Weight | 3822.44 |
订购联系方式:
上海鸿肽生物科技有限公司
手机: +86-18018095145 (同微信号)
QQ: 3259098395
邮箱:sales1@hongtide.com
本产品仅供科研使用。
关键字: L-JNKI-1;胞渗透性多肽抑制剂多肽L-JNKI-1;胞渗透性多肽抑制剂多肽;多肽;多肽合成;
上海鸿肽生物科技有限公司(简称:鸿肽生物)是一家以多肽以及多肽上下游产品研发、生产、销售以及技术转让为主要业 务科技公司。公司现有产品涵盖:定制多肽、目录多肽、氨基酸衍生物、小分子化合物;公司自成立以来,秉持“用质量作船, 以服务为帆,为科研服务”的企业理念,为国内外众多科研工作者提供了优质的服务及产品。