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111039-41-9

{[(4-bromophenyl)methyl]sulfanyl}methanimidamide hydrobromide synthesis

2synthesis methods
-

Yield:111039-41-9 97%

Reaction Conditions:

in ethanol; for 2 h;Reflux;

Steps:

7 4-Bromobenzyl Carbamimidothioate Hydrobromide

1-Bromo-4-(bromomethyl)benzene (507 mg, 2.03 mmol) and 7 thiourea (129 mg, 1.69 mmol) were dissolved in 8 ethanol (20 mL). The reaction mixture was refluxed for 2 hours. The reaction mixture was cooled, and ethanol was removed under reduced pressure. The resulting residue was suspended in dichloromethane. The suspension was filtered to give a product as a white solid (535 mg, 97%); 1H NMR (300 MHz) (DMSO-d6) δ 9.21 (s, 2H), 9.01 (s, 2H), 7.59-7.55 (m, 2H), 7.40-7.36 (m, 2H), 4.48 (s, 2H); LC/MS RT=2.406 (M+H+: 246).

References:

US2019/31624,2019,A1 Location in patent:Paragraph 0417