Welcome to chemicalbook!
Chinese English Japanese Germany Korea
400-158-6606
Try our best to find the right business for you.
Do not miss inquiry messages Please log in to view all inquiry messages.

Welcome back!

ChemicalBook CAS DataBase List 7-ALLYLOXY-4-METHYLCOUMARIN
3993-57-5

7-ALLYLOXY-4-METHYLCOUMARIN synthesis

8synthesis methods
-

Yield:3993-57-5 98%

Reaction Conditions:

in acetone;

Steps:

7-Allyloxy-4-methylcoumarin

7-Allyloxy-4-methylcoumarin 7-Hydroxy-4-methylcoumarin (70.00 g, 0.397 mol), anhydrous K2 CO3 (140 g, 1.01 mol), and allyl bromide (100 ml, 1.15 mol) were added to 2.0 L of reagent grade acetone. The milky mixture was refluxed for sixteen hours with overhead stirring, allowed to cool to room temperature, and filtered. Solids were washed once with reagent grade acetone (150 ml.), the filtrate and wash combined, and the resulting combined filtrate concentrated to dryness with a rotary evaporator to obtain 7-allyloxy-4-methylcoumarin (84.2 g, 98% yield). The crude product melted at 100.0°-101.5° C. (lit. 1 101° C.), showed only one spot in TLC, and was used in the next step.

References:

US4294847,1981,A