Welcome to chemicalbook!
Chinese English Japanese Germany Korea
400-158-6606
Try our best to find the right business for you.
Do not miss inquiry messages Please log in to view all inquiry messages.

Welcome back!

108160-14-1

Quinazoline, 4-(2-propyn-1-yloxy)- synthesis

2synthesis methods
-

Yield:108160-14-1 75%

Reaction Conditions:

Stage #1: 4-Hydroxyquinazolinewith (benzotriazo-1-yloxy)tris(dimethylamino)phosphonium hexafluorophosphate;caesium carbonate in tetrahydrofuran at 20; for 0.833333 h;Inert atmosphere;
Stage #2: propargyl alcoholwith caesium carbonate at 20; for 4 h;

References:

Kokatla, Hari Prasad;Lakshman, Mahesh K. [Organic Letters,2010,vol. 12,# 20,p. 4478 - 4481] Location in patent:supporting information; experimental part