HA-100 (hydrochloride)
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- CAS号:
- 210297-47-5
- 英文名:
- HA-100 (hydrochloride)
- 英文别名:
- HA-100 dihydrochloride
DISCONTINUED, Offer I891000;5-piperazin-1-ylsulfonylisoquinoline:dihydrochloride
- 中文名:
- HA-100 (hydrochloride)
- 中文别名:
- HA-100二盐酸盐;5-哌嗪-1-基磺酰基异喹啉:二盐酸盐
- CBNumber:
- CB53152624
- 分子式:
- C13H16ClN3O2S
- 分子量:
- 313.8
- MOL File:
- 210297-47-5.mol
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HA-100 (hydrochloride)化学性质
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储存条件:
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Store at -20°C
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溶解度:
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insoluble in EtOH; ≥131.8 mg/mL in H2O; ≥19.17 mg/mL in DMSO with ultrasonic
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形态:
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A crystalline solid
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HA-100 (hydrochloride)性质、用途与生产工艺
HA-100 dihydrochloride 是 cGMP-dependent protein kinase (PKG)、cAMP-dependent protein kinase (PKA)、protein kinase C (PKC) 和 MLC-kinase 的抑制剂，对应的IC50值分别为4 μM、8 μM、12 μM和240 μM。
| Target | Value |
PKG
(Cell-free assay)
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4 μM
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PKA
(Cell-free assay)
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8 μM
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PKC
(Cell-free assay)
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12 μM
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MLCK
(Cell-free assay)
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240 μM
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HA-100 (hydrochloride)
上下游产品信息
上游原料
下游产品
| 更新日期 | 产品编号 | 产品名称 | CAS编号 | 包装 | 价格 |
|---|
| 2024/04/30 | S2964 | HA-100 (hydrochloride)
HA-100 dihydrochloride | 210297-47-5 | 5mg | 1777.62元 |
| 2024/04/30 | S2964 | HA-100 (hydrochloride)
HA-100 dihydrochloride | 210297-47-5 | 25mg | 5315.32元 |
HA-100 (hydrochloride)
生产厂家
210297-47-5, HA-100 (hydrochloride) 相关搜索:
- 药靶配体
- 小分子
- C13H15N3O2S2HCl
- HA-100二盐酸盐
- 5-哌嗪-1-基磺酰基异喹啉:二盐酸盐
- 210297-47-5
- HA-100 dihydrochloride
DISCONTINUED, Offer I891000
- 5-piperazin-1-ylsulfonylisoquinoline:dihydrochloride