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ENPP1 Inhibitor C

ENPP1 Inhibitor C structure

CAS No.: 2378640-92-5

Chemical Name:: ENPP1 Inhibitor C

Synonyms: Enpp-1-IN-2;ENPP1 Inhibitor C;6-[(3-aminophenyl)methyl]-N,N,5-trimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine;[1,2,4]Triazolo[1,5-a]pyrimidin-7-amine, 6-[(3-aminophenyl)methyl]-N,N,5-trimethyl-

CBNumber:: CB06197878

Molecular Formula:: C15H18N6

Molecular Weight:: 282.34

MDL Number:

MOL File:: 2378640-92-5.mol

Last updated:2024-07-02 08:54:58

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ENPP1 Inhibitor C Properties

Density	1.29±0.1 g/cm3(Predicted)
storage temp.	Store at -20°C
solubility	DMF: 30 mg/ml; DMSO: 30 mg/ml; Ethanol: 30 mg/ml
form	A crystalline solid
pka	4.27±0.10(Predicted)
color	White to off-white

ENPP1 Inhibitor C Chemical Properties,Uses,Production

Description

ENPP1 inhibitor C is an inhibitor of ectonucleotide pyrophosphatase/phosphodiesterase 1 (ENPP1; IC₅₀ = 0.26 μM in a cell-free assay).¹ It is selective for ENPP1 over ENPP2-7 at 10 μM. ENPP1 inhibitor C decreases ENPP1 activity in MDA-MB-231 human breast and C6 rat glioma cancer cells when used at a concentration of 10 μM.

References

1. Kawaguchi, M., Han, X., Hisada, T., et al. Development of an ENPP1 fluorescence probe for inhibitor screening, cellular imaging, and prognostic assessment of malignant breast cancer J. Med. Chem. 62(20),9254-9269(2019).

ENPP1 Inhibitor C Preparation Products And Raw materials

Raw materials

Preparation Products

ENPP1 Inhibitor C Suppliers

Global( 11)Suppliers

Supplier	Tel	Email	Country	ProdList	Advantage
Aladdin Scientific	+1-+1(833)-552-7181	sales@aladdinsci.com	United States	52927	58
Shanghai EFE Biological Technology Co., Ltd.	021-65675885 18964387627	info@efebio.com	China	9707	58
Shenzhen SUNGENING Bio-Medical Co., Ltd.	0755-28967200 13631290199	wxf@sungening.com	China	9592	60
Shanghai Hongye Biotechnology Co. Ltd	400-9205774	sales@glpbio.cn	China	6870	58
ChemeGen(Shanghai) Biotechnology Co.,Ltd.	18818260767	sales@chemegen.com	China	11289	58
Wuhan Topule	+86-02787215551 +86-19945035818	2936752263@qq.com	China	8206	58
Xianning Shen Lan Biomedical Research and Development Co., Ltd.	18171815831	1341138380@qq.com	China	2832	58
Shanghai Tachizaki Biomedical Research Center	18014399201	sales@chemlab-tachizaki.com	China	2540	58
TargetMol Chemicals Inc.	15002134094	marketing@targetmol.cn	China	28091	58
Olix (Shanghai) Pharmaceutical Technology Co., Ltd	17316404525	209533805@qq.com	China	9718	58

Supplier	Advantage
Aladdin Scientific	58
Shanghai EFE Biological Technology Co., Ltd.	58
Shenzhen SUNGENING Bio-Medical Co., Ltd.	60
Shanghai Hongye Biotechnology Co. Ltd	58
ChemeGen(Shanghai) Biotechnology Co.,Ltd.	58
Wuhan Topule	58
Xianning Shen Lan Biomedical Research and Development Co., Ltd.	58
Shanghai Tachizaki Biomedical Research Center	58
TargetMol Chemicals Inc.	58
Olix (Shanghai) Pharmaceutical Technology Co., Ltd	58

ENPP1 Inhibitor C [1,2,4]Triazolo[1,5-a]pyrimidin-7-amine, 6-[(3-aminophenyl)methyl]-N,N,5-trimethyl- 6-[(3-aminophenyl)methyl]-N,N,5-trimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine Enpp-1-IN-2 2378640-92-5