PD 135158

CAS No.
130325-35-8
Chemical Name:
PD 135158
Synonyms
PD 135158;4-[[(1R)-2-[[(2R)-3-(1H-Indol-3-yl)-2-methyl-1-oxo-2-[[[[(1S,2R,4S)-1,7,7-trimethylbicyclo[2.2.1]hept-2-yl]oxy]carbonyl]amino]propyl]amino]-1-phenylethyl]amino]-4-oxobutanoicacid
CBNumber:
CB41400397
Molecular Formula:
C42H61N5O11
Molecular Weight:
811.97
MDL Number:
MOL File:
130325-35-8.mol
Last updated:2023-05-18 11:31:03

PD 135158 Properties

storage temp. Store at +4°C
solubility <61.68mg/ml in DMSO

PD 135158 price

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
Tocris 2608 PD135158 ≥98%(HPLC) 130325-35-8 10 $224 2021-12-16 Buy
Tocris 2608 PD135158 ≥98%(HPLC) 130325-35-8 50 $900 2021-12-16 Buy
Usbiological 256181 PD 135158 130325-35-8 10mg $559 2021-12-16 Buy
ApexBio Technology B7127 PD135158 130325-35-8 50mg $1793 2021-12-16 Buy
American Custom Chemicals Corporation API0019234 4-[[(1R)-2-[[(2R)-3-(1H-INDOL-3-YL)-2-METHYL-1-OXO-2-[[[[(1S,2R,4S)-1,7,7-TRIMETHYLBICYCLO[2.2.1]HEPT-2-YL]OXY]CARBONYL]AMINO]PROPYL]AMINO]-1-PHENYLETHYL]AMINO]-4-OXOBUTANOIC ACID 95.00% 130325-35-8 5MG $498.64 2021-12-16 Buy
Product number Packaging Price Buy
2608 10 $224 Buy
2608 50 $900 Buy
256181 10mg $559 Buy
B7127 50mg $1793 Buy
API0019234 5MG $498.64 Buy

PD 135158 Chemical Properties,Uses,Production

Biological Activity

Potent and selective, nonpeptide CCK 2 receptor antagonist (IC 50 values are 2.8 and 1232 nM for CCK 2 and CCK 1 respectively) that displays negligible affinity at GABA A , benzodiazepine, substance P, neurotensin, opioid, bradykinin and 5-HT 3 receptors (IC 50 > 10 μ M). Exhibits anxiolytic activity in elevated plus maze and social interaction tests and increases food intake in rats.

PD 135158 Preparation Products And Raw materials

Raw materials

Preparation Products

PD 135158 Suppliers

Global( 16)Suppliers
Supplier Tel Email Country ProdList Advantage
TargetMol Chemicals Inc.
+1-781-999-5354 +1-00000000000 marketing@targetmol.com United States 19892 58
3B Pharmachem (Wuhan) International Co.,Ltd. 821-50328103-801 18930552037 3bsc@sina.com China 15848 69
EMMX Biotechnology LLC 888-539-0666 info@emmx.com United States 8449 60
TargetMol Chemicals Inc. 4008200310 marketing@tsbiochem.com China 23980 58
ApexBio Technology -- sales@apexbt.com United States 6254 58
PD 135158 4-[[(1R)-2-[[(2R)-3-(1H-Indol-3-yl)-2-methyl-1-oxo-2-[[[[(1S,2R,4S)-1,7,7-trimethylbicyclo[2.2.1]hept-2-yl]oxy]carbonyl]amino]propyl]amino]-1-phenylethyl]amino]-4-oxobutanoicacid 130325-35-8