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Eptazocine

CAS No.
72150-17-5
Chemical Name:
Eptazocine
Synonyms
ST-2121;MCV 4169;l-ST-2121;(-)-ST 2121;St 2121, L-;(-)-NIH 9614;ST 2121, (-)-;Sedapain (TN);Eptazocine HBr;Eptazocine hydrobromide
CBNumber:
CB51178637
Molecular Formula:
C15H22BrNO
Molecular Weight:
312.25
MDL Number:
MFCD01714989
MOL File:
72150-17-5.mol
MSDS File:
SDS
Last updated:2024-10-23 13:36:13

Eptazocine Properties

FDA UNII 865626Y4ON

Eptazocine Chemical Properties,Uses,Production

Description

Eptazocine hydrobromide is a centrally-acting analgesic useful in the management of post-operative and cancer pain, In animal studies eptazocine exhibits a mixed agonist/antagonist profile; its analgesic activity is reported to be mediated via opiate receptors and catecholaminergic neurons.

Originator

Nichiiko (Japan)

Uses

Eptazocine Hydrobromide (CAS# 72150-17-5) can be used for various pharmaceutical compounds for improved skin penetration for opioid antagonists due to the presence of fatty acid esters and glycerin fatty acid esters.

Definition

ChEBI: Eptazocine hydrobromide is a member of tetralins.

brand name

Sedapain

Eptazocine Preparation Products And Raw materials

Raw materials

Preparation Products

(-)-NIH 9614 (-)-ST 2121 1,6-Methano-1H-4-benzazonin-10-ol, 2,3,4,5,6,7-hexahydro-1,4-dimethyl-, hydrobromide, (1S)- 1,6-Methano-1H-4-benzazonin-10-ol, 2,3,4,5,6,7-hexahydro-1,4-dimethyl-, hydrobromide, (1S,6S)- l-ST-2121 MCV 4169 ST 2121, (-)- ST-2121 (1S,6S)-2,3,4,5,6,7-Hexahydro-1,4-dimethyl-1,6-methano-1H-4-benzazepin-10-ol hydrobromide Eptazocine hydrobromide (-)-1,4-Dimethyl-10-hydroxy-2,3,4,5,6,7-hexahydro-1,6-methano-1H-4-benzazonine hydrobromide (-)-2,3,4,5,6,7-Hexahydro-1,4-dimethyl-1,6-methano-1H-4-benzazonin-10-ol hydrobromide L-1,4-Dimethyl-10-hydroxy-2,3,4,5,6,7-hexahydro-1,6-methano-1H-4-benzazonine hydrobromide St 2121, L- Sedapain (TN) Eptazocine HBr 72150-17-5