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Glucagon Receptor Antagonist, Control

CAS No.
362482-00-6
Chemical Name:
Glucagon Receptor Antagonist, Control
Synonyms
Glucagon Receptor Antagonist, Control;Glucagon Receptor Antagonist Inactive Control;4-bromo-N-[3-cyano-6-(1,1-dimethylpropyl)-4,5,6,7-tetrahydrobenzo[b]thien-2-yl]-benzamide;Benzamide, 4-bromo-N-[3-cyano-6-(1,1-dimethylpropyl)-4,5,6,7-tetrahydrobenzo[b]thien-2-yl]-;4-bromo-N-[3-cyano-6-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]benzamide
CBNumber:
CB53136787
Molecular Formula:
C21H23BrN2OS
Molecular Weight:
431.39
MDL Number:
MFCD01344061
MOL File:
362482-00-6.mol
Last updated:2023-05-21 10:59:17

Glucagon Receptor Antagonist, Control Properties

Boiling point 490.8±45.0 °C(Predicted)
Density 1.38±0.1 g/cm3(Predicted)
storage temp. Store at -20°C
solubility DMSO: Soluble
form A crystalline solid
pka 11.83±0.40(Predicted)

Glucagon Receptor Antagonist, Control price More Price(3)

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
Cayman Chemical 21188 Glucagon Receptor Antagonist Inactive Control 362482-00-6 1mg $179 2024-03-01 Buy
Cayman Chemical 21188 Glucagon Receptor Antagonist Inactive Control 362482-00-6 5mg $848 2024-03-01 Buy
AK Scientific 1374CM GlucagonReceptorAntagonist,Control 362482-00-6 1mg $322 2021-12-16 Buy
Product number Packaging Price Buy
21188 1mg $179 Buy
21188 5mg $848 Buy
1374CM 1mg $322 Buy

Glucagon Receptor Antagonist, Control Chemical Properties,Uses,Production

Description

Glucagon receptor antagonist inactive control is an analog of glucagon receptor antagonist I .1 It inhibits glucagon binding to the glucagon receptor (GCGR) by only 20% in CHO cells expressing human GCGR when used at a concentration of 10 μM. Glucagon receptor antagonist inactive control has no effect on glucagon-induced glycogenolysis in primary human hepatocytes when used at concentrations of 10 or 30 μM.

References

1. Qureshi, S.A., Candelore, M.R., Xie, D., et al. A novel glucagon receptor antagonist inhibits glucagon-mediated biological effects Diabetes 53(12),3267-3273(2004).

Glucagon Receptor Antagonist, Control Preparation Products And Raw materials

Raw materials

Preparation Products

Glucagon Receptor Antagonist, Control Suppliers

Global( 7)Suppliers
Supplier Tel Email Country ProdList Advantage
Shanghai Hongye Biotechnology Co. Ltd 400-9205774 sales@glpbio.cn China 6870 58
Shanghai Yifei Biotechnology Co. , Ltd. 021-65675885 18964387627 customer_service@efebio.com China 8740 58
TargetMol Chemicals Inc. 15002134094 marketing@targetmol.cn China 28118 58
Glucagon Receptor Antagonist, Control 4-bromo-N-[3-cyano-6-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]benzamide Glucagon Receptor Antagonist Inactive Control Benzamide, 4-bromo-N-[3-cyano-6-(1,1-dimethylpropyl)-4,5,6,7-tetrahydrobenzo[b]thien-2-yl]- 4-bromo-N-[3-cyano-6-(1,1-dimethylpropyl)-4,5,6,7-tetrahydrobenzo[b]thien-2-yl]-benzamide 362482-00-6