ChemicalBook >> CAS DataBase List >>DEBRISOQUIN SULFATE
DEBRISOQUIN SULFATE
- CAS No.
- 581-88-4
- Chemical Name:
- DEBRISOQUIN SULFATE
- Synonyms
- Tendor;declinax;RO 5-3307;RO 5-33071;Debrisoquina;Debrisochinum;ebrisoquinsulfate;DEBRISOQUIN SULFATE;DEBRISOQUINE SULFATE;isocaramidinesulfate
- CBNumber:
- CB6133940
- Molecular Formula:
- C20H28N6O4S
- Molecular Weight:
- 448.54
- MDL Number:
- MFCD00153791
- MOL File:
- 581-88-4.mol
Last updated:2024-10-23 13:36:13
| Melting point | 278-280°, 284-285° or 266-268° (H2O) |
|---|---|
| storage temp. | room temp |
| solubility | H2O: 20 mg/mL with heat |
| form | Solid |
| color | Pale Yellow |
| FDA UNII | Q94064N9NW |
DEBRISOQUIN SULFATE price More Price(16)
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| Sigma-Aldrich | D1306 | Debrisoquine sulfate | 581-88-4 | 100mg | $280 | 2024-03-01 | Buy |
| Sigma-Aldrich | BP103 | Debrisoquine sulfate British Pharmacopoeia (BP) Reference Standard | 581-88-4 | 100MG | $266 | 2024-03-01 | Buy |
| Cayman Chemical | 29568 | Debrisoquin (hemisulfate) | 581-88-4 | 10mg | $36 | 2024-03-01 | Buy |
| Cayman Chemical | 29568 | Debrisoquin (hemisulfate) | 581-88-4 | 250mg | $595 | 2024-03-01 | Buy |
| Cayman Chemical | 29568 | Debrisoquin (hemisulfate) | 581-88-4 | 50mg | $155 | 2024-03-01 | Buy |
DEBRISOQUIN SULFATE Chemical Properties,Uses,Production
Chemical Properties
Crystalline Solid
Originator
Declinax,Roche,UK,1967
Uses
Antihypertensive.
Manufacturing Process
27 g of 1,2,3,4-tetrahydroisoquinoline was added at room temperature to a
solution of 28 g of 2-methyl-2-isothiourea sulfate in 80 ml of water. The
resulting mixture was kept at room temperature with occasional shaking. After
a short period of time, methylmercaptan began to escape, and the mixture
warmed up slightly. After then standing for 24 hours, crystals formed. They
were filtered off and rinsed with ice cold water. Recrystallization from
approximately 100 ml of water yielded 1,2,3,4-tetrahydroisoquinoline-2-
carboxamidine sulfate melting at 278°C to 280°C (uncorr.).
Another batch prepared in the same manner melted at 284°C to 285°C due to
a minute difference in moisture content.
Both batches prepared above analyzed correctly for (C10H13N3)2·H2SO4.
brand name
Declinax (HoffmannLaRoche).
Therapeutic Function
Antihypertensive
Biochem/physiol Actions
Debrisoquine is an anti-hypertensive agent. It is metabolized by cytochrome P4502D6.
DEBRISOQUIN SULFATE Preparation Products And Raw materials
DEBRISOQUIN SULFATE Suppliers
Global( 34)Suppliers
| Supplier | Tel | Country | ProdList | Advantage | |
|---|---|---|---|---|---|
| Shaanxi Dideu Medichem Co. Ltd | +86-29-87569266 15319487004 | 1015@dideu.com | China | 4084 | 58 |
| TargetMol Chemicals Inc. | support@targetmol.com | United States | 38632 | 58 | |
| J & K SCIENTIFIC LTD. | 010-82848833 400-666-7788 | jkinfo@jkchemical.com | China | 96815 | 76 |
| Chemsky（shanghai）International Co.,Ltd. | 021-50135380 | shchemsky@sina.com | China | 32321 | 50 |
| Sigma-Aldrich | 021-61415566 800-8193336 | orderCN@merckgroup.com | China | 51456 | 80 |
| Shanghai EFE Biological Technology Co., Ltd. | 021-65675885 18964387627 | info@efebio.com | China | 9806 | 58 |
| Shanghai Hongye Biotechnology Co. Ltd | 400-9205774 | sales@glpbio.cn | China | 6777 | 58 |
| Shenzhen Polymeri Biochemical Technology Co., Ltd. | +86-400-002-6226 +86-13028896684; | sales@rrkchem.com | China | 57412 | 58 |
| ChemeGen(Shanghai) Biotechnology Co.,Ltd. | 18818260767 | sales@chemegen.com | China | 11217 | 58 |
| Changzhou Furuisi Biotechnology Co., Ltd | 0519-85524369 | 3477467573@qq.com | China | 8617 | 58 |
View Lastest Price from DEBRISOQUIN SULFATE manufacturers
| Image | Update time | Product | Price | Min. Order | Purity | Supply Ability | Manufacturer | |
|---|---|---|---|---|---|---|---|---|
 |
2024-10-24 | Debrisoquin sulfate
581-88-4
|
US $49.00 / mg | 10g | TargetMol Chemicals Inc. |
-
- Debrisoquin sulfate
581-88-4
- US $49.00 / mg
- TargetMol Chemicals Inc.
3,4-dihydro-2(1h)-isoquinolinecarboximidamidsulfate(2:1)
3,4-dihydro-2(1h)-isoquinolinecarboxamidinsulfate(2:1)
3,4-Dihydro-2(1H)-isoquinolinecarboximidamide, Debrisoquin sulfate, Ro5-33071
Tendor
3,4-Dihydro-2(1H)-isoquinolinecarboxamide hemisulfate
3,4-DIHYDRO-2(1H)-ISOQUINOLINECARBOXAMIDINE 0.5 H2SO4
3,4-DIHYDRO-2-[1H]-ISOQUINOLINECARBOXAMIDINE SULFATE SALT
DEBRISOQUINE SULFATE
DEBRISOQUIN SULFATE
bis(2-amidino-1,2,3,4-tetrahydroisoquinoline) sulphate
declinax
isocaramidinesulfate
RO 5-3307
RO 5-33071
2(1H)-Isoquinolinecarboximidamide, 3,4-dihydro-, sulfate (2:1)
DEBRISOQUINEHEMISULPHATE
3,4-Dihydro-2(1H)-isoquinolinecarboximidamide Hemisulfate
Debrisoquin Hemisulfate
Debrisoquine Hemisulfate
Isocaramidine Hemisulfate
3,4-dihydro-2(1h)-isoquinolinecarboxamidinesulfate
ebrisoquinsulfate
Debrisochinum
Debrisoquina
581-88-4
C10H13N32H2SO4
C20H26N6H2SO4
2C10H13N3H2O4S
C10H13N312H2SO4
Its metabolite may induce Parkinsonism.
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