FR 139317

CAS No.: 142375-60-8

Chemical Name:: FR 139317

Synonyms: FR 139317;FR139317,CID107810;N,N-hexamethylenecarbamoyl-leu-N-*methyl-D-trp-D-;(N,N-HEXAMETHYLENE) CARBAMOYL-LEU-D-TRP(N-ME)-D-2-PYA;(HEXAHYDRO-1H-AZEPINYL)CARBONYL-LEU-D-(1-ME)-TRP-DPAL;(HEXAHYDRO-1H-AZEPINYL)CARBONYL-LEU-DTRP(ME)-D-ALA(2-PYRIDYL)-OH;D-Alanine, N-((hexahydro-1H-azepin-1-yl)carbonyl)-L-leucyl-1-methyl-D-tryptophyl-3-(2-pyridinyl)-;N-[N-[N-[(HEXAHYDRO-1H-AZEPIN-1-YL)CARBONYL]-L-LEUCYL]-1-METHYL-D-TRYPTOPHYL]-3-(2-PYRIDINYL)-D-ALANINE;D-Alanine, N-(N-(N-((hexahydro-1H-azepin-1-yl)carbonyl)-L-leucyl)-1-methyl-D-tryptophyl)-3-(2-pyridinyl)-;2-((1-(Hexahydro-1H-azepinyl)carbonyl)amino-4-methylpentanoyl)-3-(-(1-methyl-1H-indolyl)propionyl)amino-3-(2-pyridyl)propionic acid

CBNumber:: CB0216568

Molecular Formula:: C33H44N6O5

Molecular Weight:: 604.74

MOL File:: 142375-60-8.mol

Modify Date:: 2024/10/23 13:36:13

Request For Quotation

FR 139317 Properties

Boiling point	943.9±65.0 °C(Predicted)
Density	1.27±0.1 g/cm3(Predicted)
storage temp.	Desiccate at +4°C
solubility	Soluble to 100 mM in 1eq. HCl and to 100 mM in DMSO
form	Powder
pka	2.68±0.10(Predicted)

FR 139317 Chemical Properties,Uses,Production

Uses

FR 139317 is a novel, potent endothelin ETA receptor antagonist.

Biological Activity

A highly potent and selective ET A endothelin receptor antagonist (K i values are 1 nM and 7.3 μ M at ET A and ET B subtypes respectively). Active in vivo .

FR 139317 Preparation Products And Raw materials

Raw materials

Preparation Products

FR 139317 Suppliers

Global( 41)Suppliers

Supplier	Tel	Country	ProdList	Advantage	Inquiry
TargetMol Chemicals Inc.	+1-781-999-5354 +1-00000000000	United States	32080	58	Inquiry
Zhejiang J&C Biological Technology Co.,Limited	+1-2135480471 +1-2135480471	China	10473	58	Inquiry
Aladdin Scientific	+1-+1(833)-552-7181	United States	57505	58	Inquiry
TargetMol Chemicals Inc.	+8613564774135	United States	19863	58	Inquiry
Hangzhou Sinoda Pharmaceutical Technology Co. LTD	0571-87213919 17306812703	China	6445	58	Inquiry
Zhongke Huayao (Jiangsu) Biotechnology Co., Ltd	18014456767	China	1350	58	Inquiry
Shanghai Aladdin Biochemical Technology Co.,Ltd.	+86-18521732826	China	48461	58	Inquiry
Jiangsu Aikon Biopharmaceutical R&D Co.,Ltd.	025-66061636 18013972705	China	10238	58	Inquiry
TargetMol Chemicals Inc.	4008200310	China	24647	58	Inquiry
Alexis Corporation	+41 61 926 8989	Switzerland	3599	74	Inquiry

Supplier	Advantage
TargetMol Chemicals Inc.	58
Zhejiang J&C Biological Technology Co.,Limited	58
Aladdin Scientific	58
TargetMol Chemicals Inc.	58
Hangzhou Sinoda Pharmaceutical Technology Co. LTD	58
Zhongke Huayao (Jiangsu) Biotechnology Co., Ltd	58
Shanghai Aladdin Biochemical Technology Co.,Ltd.	58
Jiangsu Aikon Biopharmaceutical R&D Co.,Ltd.	58
TargetMol Chemicals Inc.	58
Alexis Corporation	74

FR 139317 Spectrum

FR 139317(142375-60-8)MS FR 139317(142375-60-8)IR1

142375-60-8(FR 139317)Related Search:

3-(2-Pyridyl)-D-alanine BETA-(2-PYRIDYL)-DL-ALANINE 2-Pyridinepropanol 3-PYRIDIN-2-YL-PROPIONIC ACID H2SO4 FR 139317

2-(2-Methoxyphenoxy)ethylamine 1-METHYL-2-PYRIDIN-2-YL-ETHYLAMINE N-ACETYL-D-ALA-D-ALA 1H-Azepine-1-carboxamide,hexahydro-(9CI) METHYL-(1-METHYL-2-PYRIDIN-2-YL-ETHYL)-AMINE

chevron_left

1of2

chevron_right

FR 139317 (HEXAHYDRO-1H-AZEPINYL)CARBONYL-LEU-D-(1-ME)-TRP-DPAL (HEXAHYDRO-1H-AZEPINYL)CARBONYL-LEU-DTRP(ME)-D-ALA(2-PYRIDYL)-OH 2-((1-(Hexahydro-1H-azepinyl)carbonyl)amino-4-methylpentanoyl)-3-(-(1-methyl-1H-indolyl)propionyl)amino-3-(2-pyridyl)propionic acid D-Alanine, N-((hexahydro-1H-azepin-1-yl)carbonyl)-L-leucyl-1-methyl-D-tryptophyl-3-(2-pyridinyl)- D-Alanine, N-(N-(N-((hexahydro-1H-azepin-1-yl)carbonyl)-L-leucyl)-1-methyl-D-tryptophyl)-3-(2-pyridinyl)- N-[N-[N-[(HEXAHYDRO-1H-AZEPIN-1-YL)CARBONYL]-L-LEUCYL]-1-METHYL-D-TRYPTOPHYL]-3-(2-PYRIDINYL)-D-ALANINE (N,N-HEXAMETHYLENE) CARBAMOYL-LEU-D-TRP(N-ME)-D-2-PYA N,N-hexamethylenecarbamoyl-leu-N-*methyl-D-trp-D- FR139317,CID107810 (2R)-2-[[(2R)-2-[[(2S)-2-(AZEPANE-1-CARBONYLAMINO)-4-METHYLPENTANOYL]AMINO]-3-(1-METHYLINDOL-3-YL)PROPANOYL]AMINO]-3-PYRIDIN-2-YLPROPANOIC ACID 142375-60-8 C33H44N6O5