MRS 2279
- CAS No.
- 367909-40-8
- Chemical Name:
- MRS 2279
- Synonyms
- MRS 2279;MRS2279,MRS-2279;MRS 2279, CID: 5311301;[(1S,2R,4R)-4-[(2-chloro-6-methylaminopurin-9-yl)methyl]-2-(phosphonooxymethyl)cyclopentyl] dihydrogen phosphate;Bicyclo[3.1.0]hexane-1-methanol, 4-[2-chloro-6-(methylamino)-9H-purin-9-yl]-2-(phosphonooxy)-, 1-(dihydrogen phosphate), (1R,2S,4S,5S)-;(1R*,2S*)-4-[2-Chloro-6-(methylamino)-9H-purin-9-yl]-2-(phosphonooxy)bicyclo[3.1.0]hexane-1-methanoldihydrogenphosphateesterdiammoniumsalt
- CBNumber:
- CB3848748
- Molecular Formula:
- C13H18ClN5O8P2
- Molecular Weight:
- 469.71
- MOL File:
- 367909-40-8.mol
- Modify Date:
- 2023/5/18 11:31:02
MRS 2279 Chemical Properties,Uses,Production
Uses
MRS 2279 is a selective P2Y1 antagonist with high affinity and results in modulation of aggregation of blood platelets induced by ADP.
Biological Activity
Selective, high affinity competitive antagonist of the P2Y 1 receptor (K i = 2.5 nM; IC 50 = 51.6 nM). Fails to block nucleotide signaling at most other P2Y receptors (P2Y 2 , P2Y 4 , P2Y 6 , P2Y 11 and P2Y 12 ) and potently inhibits ADP-induced aggregation of human blood platelets in vitro (pK B = 8.05).
MRS 2279 Preparation Products And Raw materials
Raw materials
Preparation Products
MRS 2279 Suppliers
Global( 19)Suppliers
Supplier | Tel | Country | ProdList | Advantage | Inquiry |
---|---|---|---|---|---|
TargetMol Chemicals Inc. | +1-781-999-5354 +1-00000000000 | United States | 19892 | 58 | Inquiry |
Hangzhou MolCore BioPharmatech Co.,Ltd. | +86-057181025280; +8617767106207 | China | 49739 | 58 | Inquiry |
TargetMol Chemicals Inc. | 4008200310 | China | 23962 | 58 | Inquiry |
BOC Sciences | USA | 0 | 65 | Inquiry | |
Service Chemical Inc. | 888-895-6920 | Germany | 6373 | 71 | Inquiry |
3B Pharmachem (Wuhan) International Co.,Ltd. | 821-50328103-801 18930552037 | China | 15848 | 69 | Inquiry |
Tocris Bioscience | +44 (0) 117 916 3333 | United Kingdom | 5729 | 77 | Inquiry |
ApexBio Technology | + 1-832-696-8203 | United States | 6254 | 58 | Inquiry |
Beijing Bolide Biotechnology Co., Ltd. | 010-51653916 | CHINA | 6172 | 58 | Inquiry |
Shanghai Chaoyan Biotechnology Co., Ltd. | 021-50840550 | CHINA | 6217 | 58 | Inquiry |
367909-40-8(MRS 2279)Related Search:
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MRS 2279
(1R*,2S*)-4-[2-Chloro-6-(methylamino)-9H-purin-9-yl]-2-(phosphonooxy)bicyclo[3.1.0]hexane-1-methanoldihydrogenphosphateesterdiammoniumsalt
[(1S,2R,4R)-4-[(2-chloro-6-methylaminopurin-9-yl)methyl]-2-(phosphonooxymethyl)cyclopentyl] dihydrogen phosphate
MRS 2279, CID: 5311301
Bicyclo[3.1.0]hexane-1-methanol, 4-[2-chloro-6-(methylamino)-9H-purin-9-yl]-2-(phosphonooxy)-, 1-(dihydrogen phosphate), (1R,2S,4S,5S)-
MRS2279,MRS-2279
367909-40-8
C13H18ClN5O8P22NH3
C13H18ClN5O8P2