(R)-AM1241

(R)-AM1241 価格

メーカー	製品番号	製品説明	CAS番号	包装	価格	更新時間	購入

(R)-AM1241 化学特性,用途語,生産方法

説明

(R)-AM1241 binds to cannabinoid (CB) receptors and has greater than 100-fold selectivity for the CB₂ over the CB₁ receptor (K_is = 15 and 5,000 nM, respectively, in a membrane assay using human receptors). (R)-AM1241 acts as an agonist at human CB₂ receptors (EC₅₀ = 118 nM) but an inverse agonist at rat and mouse CB₂ receptors (EC₅₀s = 315 and 341 nM, respectively). Similar to the racemate AM1241 , (R)-AM1241 produces antinociception to thermal, but not mechanical, pain in rats. The pain-reducing effect of (R)-AM1241 is blocked by the CB₂-specific inhibitor SR 144528 but not by either the CB₁-selective inhibitor rimonabant or the opioid receptor blocker naloxone ( | ISO60191).

(R)-AM1241 上流と下流の製品情報

原材料

準備製品

(R)-AM1241 生産企業

名前	電話番号	電子メール	国籍	製品カタログ	優位度
Shanghai Hongye Biotechnology Co. Ltd	400-9205774	sales@glpbio.cn	China	6777	58

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• 444912-51-0
• (R)-AM1241
• ZUHIXXCLLBMBDW-MRXNPFEDSA-N
• (R)-AM1241 Exclusive
• (R) AM1241,(R)-AM-1241,(R)AM1241
• Methanone, (2-iodo-5-nitrophenyl)[1-[[(2R)-1-methyl-2-piperidinyl]methyl]-1H-indol-3-yl]-