バレスプラジブ 化学特性,用途語,生産方法
溶解性
In vitro (25℃) DMSO 76 mg/mL (199.79 mM)
効能
脂質異常症治療薬, 分泌型ホスホリパーゼ阻害薬
使用
VARESPLADIB is used as a PLA2 inhibitor (Phospholipase A2 Enzyme inhibitor).
Biochem/physiol Actions
Varespladib is effective against viper and elapid venoms and is used in snakebite therapy. It is reported to interact with the hydrophobic channel of the PLA2-like toxin in in vitro structural studies. It blocks inflammatory cascades related to the sPLA2.
バレスプラジブ 上流と下流の製品情報
原材料
準備製品