타비모렐린

타비모렐린
타비모렐린 구조식 이미지
카스 번호:
193079-69-5
한글명:
타비모렐린
동의어(한글):
타비모렐린
상품명:
Tabimorelin
동의어(영문):
NNC260703;NNC-260703;NNC26-0703;NNC-26-0703;Tabimorelin;Unii-L51cbe03kf;Tabimorelin [inn];N-[5-Amino-5-Methyl-2(E)-Hexenoyl]-N-Methyl-3-(2- Naphthyl)-D-Alanyl-N-Methyl-D-Phenylalanine Methylamide;D-Phenylalaninamide, N-[(2E)-5-amino-5-methyl-1-oxo-2-hexen-1-yl]-N-methyl-3-(2-naphthalenyl)-D-alanyl-N,Nα-dimethyl-;N-[(2E)-5-Amino-5-methyl-1-oxo-2-hexenyl]-N-methyl-3-(2-naphthalenyl)-D-alanyl-N,Nα-dimethyl-D-phenylalaninamidehemifumarate
CBNumber:
CB31074328
분자식:
C32H40N4O3
포뮬러 무게:
528.68
MOL 파일:
193079-69-5.mol

타비모렐린 속성

녹는점
>70°C(dec.)
끓는 점
794.4±60.0 °C(Predicted)
밀도
1.146±0.06 g/cm3(Predicted)
저장 조건
Desiccate at RT
용해도
클로로포름(약간 용해됨), DMSO(약간 용해됨), 메탄올(약간 용해됨)
산도 계수 (pKa)
15.14±0.46(Predicted)
물리적 상태
고체
물리적 상태
단단한 모양
색상
흰색에서 황백색까지
안정성
감광성

안전

타비모렐린 C화학적 특성, 용도, 생산

용도

NN703 (Tabimorelin) is an orally active growth hormone (GH) secretagogue intended for use as an alternative to daily injections of GH. In vitro studies in human liver microsomes have indicated that NN703 is a mechanism-based inhibitor of CYP3A4.

생물학적 활성

Potent, orally active ghrelin receptor (GHS-R1a) agonist (K i = 50 nM at human recombinant GHS-R1a). Stimulates GH release from rat pituitary cells with an EC 50 value of 2.7 nM. Induces hyperphagia and adiposity in lean rats, but not in leptin signaling-deficient ZDF rats.

타비모렐린 준비 용품 및 원자재

원자재

준비 용품


타비모렐린 공급 업체

글로벌( 21)공급 업체
공급자 전화 이메일 국가 제품 수 이점
3B Pharmachem (Wuhan) International Co.,Ltd. 821-50328103-801 18930552037
3bsc@sina.com China 15848 69
Chemsky (shanghai) International Co.,Ltd 021-50135380
shchemsky@sina.com China 15421 60
Beijing HuaMeiHuLiBiological Chemical 010-56205725
waley188@sohu.com China 12338 58
EMMX Biotechnology LLC 888-539-0666
info@emmx.com United States 8449 60
Hangzhou Peptidego Biotech Co.,Ltd. 0571-87213919
eric@peptidego.com China 6757 58
Jiangsu Hongmin Pharmaceutical Co., Ltd. 18221292452
fannieliu@glschina.com China 6799 58
Hangzhou Sinoda Pharmaceutical Technology Co. LTD 0571-87213919 17306812703
3007955328@qq.com China 6445 58
LGC Science (Shanghai) Ltd. 17717235263
cindy.yang@lgcgroup.com China 11677 58
Hubei Qingbei Yunyan Pharmaceutical Technology Co., Ltd 18162595016; 18162595016
3287908757@qq.com China 9117 58

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