4-(1H-IMIDAZOL-4-YLMETHYL)-1-METHYLPIPERIDINE DIHYDROBROMIDE C화학적 특성, 용도, 생산
용도
4-(1H-Imidazol-4-ylmethyl)-1-methylpiperidine Dihydrobromide is a salt analog of methimepip, which exhibits high affinity and agonist activity at the human histamine H3 receptor.
생물학적 활성
Extremely selective histamine H 3 receptor agonist (pK i values are 9.0, 5.7, < 5.0 and < 5.0 for hH 3 , hH 4 , hH 1 and hH 2 receptors respectively). Potently inhibits EFS-evoked contractions of guinea pig ileum (pD 2 = 8.26).
4-(1H-IMIDAZOL-4-YLMETHYL)-1-METHYLPIPERIDINE DIHYDROBROMIDE 준비 용품 및 원자재
원자재
준비 용품
4-(1H-IMIDAZOL-4-YLMETHYL)-1-METHYLPIPERIDINE DIHYDROBROMIDE 공급 업체