GW311616A
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GW311616A 속성
- 저장 조건
- 2-8°C
- 용해도
- H2O: 24 mg/mL, 가용성
- 물리적 상태
- 고체
- 물리적 상태
- 단단한 모양
- 색상
- White to yellow
안전
- 위험 및 안전 성명
- 위험 및 사전주의 사항 (GHS)
GW311616A C화학적 특성, 용도, 생산
개요
GW 311616A is an inhibitor of neutrophil elastase (IC50 = 100 nM). It is selective for neutrophil elastase (IC50 = 22 nM for the human enzyme) over trypsin, cathepsin G, and plasmin (IC50s = >100 μM for all), as well as chymotrypsin and tissue plasminogen activator (IC50s = >3 μM for both), in cell-free assays. GW 311616A (20 μM) inhibits the formation of neutrophil extracellular traps (NETs) induced by phorbol 12-myristate 13-acetate (PMA; ) in isolated human neutrophils. It inhibits intraneutrophil elastase activity in isolated dog blood six hours after administration of a 0.22 mg/kg dose. GW 311616A also inhibits neutrophil elastase in the liver in a mouse model of liver ischemia-reperfusion injury when administered at a dose of 2 mg/kg.GW311616A 준비 용품 및 원자재
원자재
준비 용품
GW311616A 공급 업체
글로벌( 26)공급 업체
공급자 | 전화 | 이메일 | 국가 | 제품 수 | 이점 |
---|---|---|---|---|---|
TargetMol Chemicals Inc. | +1-781-999-5354 +1-00000000000 |
marketing@targetmol.com | United States | 31974 | 58 |
Hangzhou MolCore BioPharmatech Co.,Ltd. | +86-057181025280; +8617767106207 |
sales@molcore.com | China | 49734 | 58 |
TargetMol Chemicals Inc. | |
support@targetmol.com | United States | 38459 | 58 |
Amadis Chemical Company Limited | 571-89925085 |
sales@amadischem.com | China | 131957 | 58 |
ShangHai KenEn Chemical Technology Co., Ltd. | 13120367189 |
mychess007@163.com | China | 1994 | 55 |
SPIRO PHARMA | |
eric_feng1954@126.com | China | 9248 | 55 |
BOC Sciences | 16314854226 |
info@bocsci.com | United States | 9923 | 65 |
Shanghai EFE Biological Technology Co., Ltd. | 021-65675885 18964387627 |
info@efebio.com | China | 9806 | 58 |
Musechem | +1-800-259-7612 |
info@musechem.com | United States | 4660 | 60 |
DC Chemicals | 021-58447131 13564518121 |
sales@dcchemicals.com | China | 9410 | 58 |