3-(3,5-Dibromo-4-hydroxybenzoyl)-2-ethyl-N-[4-[(2-thiazolylamino)sulfonyl]phenyl]-6-benzofuransulfonamide
![3-(3,5-Dibromo-4-hydroxybenzoyl)-2-ethyl-N-[4-[(2-thiazolylamino)sulfonyl]phenyl]-6-benzofuransulfonamide price.](/CAS2/GIF/765317-72-4.gif)
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- $61 - $479
- Product name: 3-(3,5-Dibromo-4-hydroxybenzoyl)-2-ethyl-N-[4-[(2-thiazolylamino)sulfonyl]phenyl]-6-benzofuransulfonamide
- CAS: 765317-72-4
- MF: C26H19Br2N3O7S3
- MW: 741.45
- EINECS:
- MDL Number:MFCD09037556
- Synonyms:3-(3,5-Dibromo-4-hydroxybenzoyl)-2-ethyl-N-[4-[(2-thiazolylamino)sulfonyl]phenyl]-6-benzofuransulfonamide;6-BenzofuransulfonaMide, 3-(3,5-dibroMo-4-hydroxybenzoyl)-2-ethyl-N-[4-[(2-thiazolylaMino)sulfonyl]phenyl]-;3-(3,5-Dibromo-4-hydroxybenzoyl)-2-ethyl-N-[4-(1,3-thiazol-2-ylsulfamoyl)phenyl]-1-benzofuran-6-sulfonamide;PTP1B-IN-4;PTP1B Inhibitor inhibitor
7 prices
Selected condition：
Brand
- Alfa Aesar
- Cayman Chemical
- Sigma-Aldrich
- TRC
Package
- 500μg
- 1mg
- 5mg
- 10mg
- ManufacturerAlfa Aesar
- Product numberJ64512
- Product descriptionPTP1B Inhibitor
- Packaging5mg
- Price$479
- Updated2023-06-20
- Buy
- ManufacturerCayman Chemical
- Product number15782
- Product descriptionPTP1B Inhibitor ≥98%
- Packaging500μg
- Price$61
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number15782
- Product descriptionPTP1B Inhibitor ≥98%
- Packaging1mg
- Price$112
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number15782
- Product descriptionPTP1B Inhibitor ≥98%
- Packaging5mg
- Price$264
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number15782
- Product descriptionPTP1B Inhibitor ≥98%
- Packaging10mg
- Price$468
- Updated2024-03-01
- Buy
- ManufacturerSigma-Aldrich
- Product number539741
- Product descriptionPTP1B Inhibitor - CAS 765317-72-4 - Calbiochem PTP1B Inhibitor, CAS 765317-72-4, is a cell-permeable, selective, reversible and non-competitive allosteric inhibitor of PTP1B (IC?? = 4 μM and 8 μM for PTP1B403 and PTP1B298, respectively).
- Packaging5MG
- Price$280
- Updated2023-06-20
- Buy
- ManufacturerTRC
- Product numberD421300
- Product description3-(3,5-Dibromo-4-hydroxybenzoyl)-2-ethyl-N-[4-(1,3-thiazol-2-ylsulfamoyl)phenyl]-1-benzofuran-6-sulfonamide
- Packaging1mg
- Price$100
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| Alfa Aesar | J64512 | PTP1B Inhibitor | 5mg | $479 | 2023-06-20 | Buy |
| Cayman Chemical | 15782 | PTP1B Inhibitor ≥98% | 500μg | $61 | 2024-03-01 | Buy |
| Cayman Chemical | 15782 | PTP1B Inhibitor ≥98% | 1mg | $112 | 2024-03-01 | Buy |
| Cayman Chemical | 15782 | PTP1B Inhibitor ≥98% | 5mg | $264 | 2024-03-01 | Buy |
| Cayman Chemical | 15782 | PTP1B Inhibitor ≥98% | 10mg | $468 | 2024-03-01 | Buy |
| Sigma-Aldrich | 539741 | PTP1B Inhibitor - CAS 765317-72-4 - Calbiochem PTP1B Inhibitor, CAS 765317-72-4, is a cell-permeable, selective, reversible and non-competitive allosteric inhibitor of PTP1B (IC?? = 4 μM and 8 μM for PTP1B403 and PTP1B298, respectively). | 5MG | $280 | 2023-06-20 | Buy |
| TRC | D421300 | 3-(3,5-Dibromo-4-hydroxybenzoyl)-2-ethyl-N-[4-(1,3-thiazol-2-ylsulfamoyl)phenyl]-1-benzofuran-6-sulfonamide | 1mg | $100 | 2021-12-16 | Buy |
Properties
Boiling point :855.0±75.0 °C(Predicted)
Density :1.812±0.06 g/cm3(Predicted)
storage temp. :Store at -20°C, protect from light
solubility :Soluble in ethanol and DMSO
pka :4.47±0.25(Predicted)
form :Solid
color :White to off-white
Sensitive :Light Sensitive
Density :1.812±0.06 g/cm3(Predicted)
storage temp. :Store at -20°C, protect from light
solubility :Soluble in ethanol and DMSO
pka :4.47±0.25(Predicted)
form :Solid
color :White to off-white
Sensitive :Light Sensitive
Safety Information
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Description
Protein tyrosine phosphatase 1B (PTP1B) has critical roles in cell signaling relevant to diabetes, obesity, and cancer. PTP1B inhibitor is a cell-permeable allosteric inhibitor of PTP1B (IC50s = 4 and 8 μM for 403 and 298 residue PTP1B forms, respectively). It binds reversibly and non-competitively, altering the conformation of the catalytic pocket. PTP1B inhibitor selectively increases the phosphorylation of the insulin receptor, insulin receptor substrate 1, and Akt, mimicking the action of insulin.Suppliers and manufacturers
Alchem Pharmtech,Inc.
TargetMol Chemicals Inc.
Nantong HI-FUTURE Biology Co., Ltd.
Wuhan Topule Biopharmaceutical Co., Ltd
Shenyang Zhongshen Zekang Biomedical Technology Research Co., Ltd
Aladdin Scientific
Wuhan Jingkang en Biomedical Technology Co., Ltd
Amadis Chemical Company Limited
VDM Biochemicals
China Langchem Inc.