CAY10618
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- $20 - $383
- Product name: CAY10618
- CAS: 1202580-59-3
- MF: C27H29N5O
- MW: 439.55
- EINECS:
- MDL Number:
- Synonyms:CAY10618;1H-1,2,3-Triazole-1-octanaMide, N-[1,1'-biphenyl]-2-yl-4-(3-pyridinyl)-;GPP 78;CAY10618 Exclusive;N-(2-phenylphenyl)-8-(4-pyridin-3-yltriazol-1-yl)octanamide;GPP78,GPP-78
6 prices
Selected condition：
Brand
- AK Scientific
- Cayman Chemical
Package
- 500μg
- 1mg
- 5mg
- 10mg
- ManufacturerAK Scientific
- Product number4481DF
- Product descriptionN-(2-Phenylphenyl)-8-[4-(3-pyridinyl)-1-triazolyl]octanamide
- Packaging5mg
- Price$262
- Updated2021-12-16
- Buy
- ManufacturerAK Scientific
- Product number4481DF
- Product descriptionN-(2-Phenylphenyl)-8-[4-(3-pyridinyl)-1-triazolyl]octanamide
- Packaging10mg
- Price$383
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number13670
- Product descriptionGPP 78 ≥95%
- Packaging500μg
- Price$20
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number13670
- Product descriptionGPP 78 ≥95%
- Packaging1mg
- Price$37
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number13670
- Product descriptionGPP 78 ≥95%
- Packaging5mg
- Price$146
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number13670
- Product descriptionGPP 78 ≥95%
- Packaging10mg
- Price$257
- Updated2024-03-01
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| AK Scientific | 4481DF | N-(2-Phenylphenyl)-8-[4-(3-pyridinyl)-1-triazolyl]octanamide | 5mg | $262 | 2021-12-16 | Buy |
| AK Scientific | 4481DF | N-(2-Phenylphenyl)-8-[4-(3-pyridinyl)-1-triazolyl]octanamide | 10mg | $383 | 2021-12-16 | Buy |
| Cayman Chemical | 13670 | GPP 78 ≥95% | 500μg | $20 | 2024-03-01 | Buy |
| Cayman Chemical | 13670 | GPP 78 ≥95% | 1mg | $37 | 2024-03-01 | Buy |
| Cayman Chemical | 13670 | GPP 78 ≥95% | 5mg | $146 | 2024-03-01 | Buy |
| Cayman Chemical | 13670 | GPP 78 ≥95% | 10mg | $257 | 2024-03-01 | Buy |
Properties
Density :1.15±0.1 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :DMF: 10 mg/ml; DMSO: 10 mg/ml; DMSO:PBS(pH 7.2) (1:3): 0.25 mg/ml; Ethanol: 10 mg/ml
pka :14.80±0.70(Predicted)
form :Liquid
color :Colorless to light yellow
storage temp. :Store at -20°C
solubility :DMF: 10 mg/ml; DMSO: 10 mg/ml; DMSO:PBS(pH 7.2) (1:3): 0.25 mg/ml; Ethanol: 10 mg/ml
pka :14.80±0.70(Predicted)
form :Liquid
color :Colorless to light yellow
Safety Information
| Symbol(GHS): |
 
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| Signal word: | Danger | |||||||
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Description
Nicotinamide phosphoribosyltransferase (Nampt) converts nicotinamide into nicotinamide mononucleotide (NMN), which is subsequently converted to NAD+ by NMN adenyltransferase. Cancer cells commonly have an unusually high rate of NAD+ turnover, suggesting that inhibition of Nampt might selectively target cancer cells. ?GPP 78 is a potent inhibitor of Nampt (IC50 = 3 nM). It induces cell death in the neuroblastoma cell line SH-SY5Y with an IC50 value of 3.8 nM through a process that appears to involve autophagy.Suppliers and manufacturers
TargetMol Chemicals Inc.
BOC Sciences
Beijing Jin Ming Biotechnology Co., Ltd.
Shanghai Hongye Biotechnology Co. Ltd
Chengdu Peter-like Biotechnology Co., Ltd.
ChemeGen(Shanghai) Biotechnology Co.,Ltd.
Beijing Jin Ming Biotechnology Co., Ltd.
TargetMol Chemicals Inc.
Shanghai Yifei Biotechnology Co. , Ltd.