PKI-402
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- $57 - $2986.9
- Product name: PKI-402
- CAS: 1173204-81-3
- MF: C29H34N10O3
- MW: 570.65
- EINECS:
- MDL Number:MFCD18251484
- Synonyms:1-(4-(3-ethyl-7-morpholino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl)phenyl)-3-(4-(1-methylpiperazine-4-carbonyl)phenyl)urea;1-(4-(3-ethyl-7-morpholino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl)phenyl)-3-(4-(4-methylpiperazine-1-carbonyl)phenyl)urea;PKI-402;PKI402;1-(4-(3-Ethyl-7-morpholino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl)phenyl)-3-(4-(4-methylpiper;PKI-402;1-[4-[3-Ethyl-7-(morpholin-4-yl)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl]phenyl]-3-[4-[(4-methylpiperazin-1-yl)carbonyl]phenyl]urea;CS-167;Urea, N-[4-[3-ethyl-7-(4-morpholinyl)-3H-1,2,3-triazolo[4,5-d]pyrimidin-5-yl]phenyl]-N'-[4-[(4-methyl-1-piperazinyl)carbonyl]phenyl]-
29 prices
Selected condition:
Brand
- AK Scientific
- American Custom Chemicals Corporation
- ApexBio Technology
- Biorbyt Ltd
- Cayman Chemical
- ChemScene
- Crysdot
- DC Chemicals
- Medical Isotopes, Inc.
- TRC
Package
- 50mg
- 100mg
- 250mg
- 1000mg
- 10mM(in 1mL DMSO)
- 1mg
- 5MG
- 10mg
- 25MG
- ManufacturerAK Scientific
- Product numberY0339
- Product description1-(4-(3-ethyl-7-morpholino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl)phenyl)-3-(4-(1-methylpiperazine-4-carbonyl)phenyl)urea
- Packaging1mg
- Price$160
- Updated2021-12-16
- Buy
- ManufacturerAK Scientific
- Product numberY0339
- Product description1-(4-(3-ethyl-7-morpholino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl)phenyl)-3-(4-(1-methylpiperazine-4-carbonyl)phenyl)urea
- Packaging10mg
- Price$586
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberKIN0001407
- Product description1-[4-[3-ETHYL-7-(MORPHOLIN-4-YL)-3H-[1,2,3]TRIAZOLO[4,5-D]PYRIMIDIN-5-YL]PHENYL]-3-[4-[(4-METHYLPIPERAZIN-1-YL)CARBONYL]PHENYL]UREA 95.00%
- Packaging5MG
- Price$381.7
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberKIN0001407
- Product description1-[4-[3-ETHYL-7-(MORPHOLIN-4-YL)-3H-[1,2,3]TRIAZOLO[4,5-D]PYRIMIDIN-5-YL]PHENYL]-3-[4-[(4-METHYLPIPERAZIN-1-YL)CARBONYL]PHENYL]UREA 95.00%
- Packaging25MG
- Price$1328.25
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA8505
- Product descriptionPKI-402
- Packaging5mg
- Price$149
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA8505
- Product descriptionPKI-402
- Packaging10mg
- Price$259
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA8505
- Product descriptionPKI-402
- Packaging10mM(in 1mL DMSO)
- Price$270
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA8505
- Product descriptionPKI-402
- Packaging50mg
- Price$679
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb180983
- Product descriptionPKI402 >98%
- Packaging100mg
- Price$765
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb180983
- Product descriptionPKI402 >98%
- Packaging250mg
- Price$1504.5
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb180983
- Product descriptionPKI402 >98%
- Packaging1000mg
- Price$2986.9
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number27664
- Product descriptionPKI-402
- Packaging1mg
- Price$57
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number27664
- Product descriptionPKI-402
- Packaging5mg
- Price$233
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number27664
- Product descriptionPKI-402
- Packaging10mg
- Price$437
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number27664
- Product descriptionPKI-402
- Packaging25mg
- Price$957
- Updated2024-03-01
- Buy
- ManufacturerChemScene
- Product numberCS-0565
- Product descriptionPKI-402 99.79%
- Packaging5mg
- Price$198
- Updated2021-12-16
- Buy
Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
---|---|---|---|---|---|---|
AK Scientific | Y0339 | 1-(4-(3-ethyl-7-morpholino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl)phenyl)-3-(4-(1-methylpiperazine-4-carbonyl)phenyl)urea | 1mg | $160 | 2021-12-16 | Buy |
AK Scientific | Y0339 | 1-(4-(3-ethyl-7-morpholino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl)phenyl)-3-(4-(1-methylpiperazine-4-carbonyl)phenyl)urea | 10mg | $586 | 2021-12-16 | Buy |
American Custom Chemicals Corporation | KIN0001407 | 1-[4-[3-ETHYL-7-(MORPHOLIN-4-YL)-3H-[1,2,3]TRIAZOLO[4,5-D]PYRIMIDIN-5-YL]PHENYL]-3-[4-[(4-METHYLPIPERAZIN-1-YL)CARBONYL]PHENYL]UREA 95.00% | 5MG | $381.7 | 2021-12-16 | Buy |
American Custom Chemicals Corporation | KIN0001407 | 1-[4-[3-ETHYL-7-(MORPHOLIN-4-YL)-3H-[1,2,3]TRIAZOLO[4,5-D]PYRIMIDIN-5-YL]PHENYL]-3-[4-[(4-METHYLPIPERAZIN-1-YL)CARBONYL]PHENYL]UREA 95.00% | 25MG | $1328.25 | 2021-12-16 | Buy |
ApexBio Technology | A8505 | PKI-402 | 5mg | $149 | 2021-12-16 | Buy |
ApexBio Technology | A8505 | PKI-402 | 10mg | $259 | 2021-12-16 | Buy |
ApexBio Technology | A8505 | PKI-402 | 10mM(in 1mL DMSO) | $270 | 2021-12-16 | Buy |
ApexBio Technology | A8505 | PKI-402 | 50mg | $679 | 2021-12-16 | Buy |
Biorbyt Ltd | orb180983 | PKI402 >98% | 100mg | $765 | 2021-12-16 | Buy |
Biorbyt Ltd | orb180983 | PKI402 >98% | 250mg | $1504.5 | 2021-12-16 | Buy |
Biorbyt Ltd | orb180983 | PKI402 >98% | 1000mg | $2986.9 | 2021-12-16 | Buy |
Cayman Chemical | 27664 | PKI-402 | 1mg | $57 | 2024-03-01 | Buy |
Cayman Chemical | 27664 | PKI-402 | 5mg | $233 | 2024-03-01 | Buy |
Cayman Chemical | 27664 | PKI-402 | 10mg | $437 | 2024-03-01 | Buy |
Cayman Chemical | 27664 | PKI-402 | 25mg | $957 | 2024-03-01 | Buy |
ChemScene | CS-0565 | PKI-402 99.79% | 5mg | $198 | 2021-12-16 | Buy |
Properties
Boiling point :670.6±55.0 °C(Predicted)
Density :1.43
storage temp. :Store at -20°C
solubility :insoluble in EtOH; insoluble in H2O; ≥14.28 mg/mL in DMSO
form :solid
pka :13.80±0.70(Predicted)
color :White to off-white
Density :1.43
storage temp. :Store at -20°C
solubility :insoluble in EtOH; insoluble in H2O; ≥14.28 mg/mL in DMSO
form :solid
pka :13.80±0.70(Predicted)
color :White to off-white
Safety Information
Symbol(GHS): |
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Signal word: | Warning | |||||||||||||||||||||
Hazard statements: |
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Description
A selective, reversible and ATP-competitive Class I PI3K inhibitor. PI3Kα, IC50=1 nM; PI3Kβ, IC50=7 nM; PI3Kγ, IC50=16 nM; PI3Kδ, IC50=14 nM.More related product prices
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