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ChemicalBook >> CAS DataBase List >> (R)-AM1241

(R)-AM1241

(R)-AM1241 price.
  • $63 - $1281
  • Product name: (R)-AM1241
  • CAS: 444912-51-0
  • MF: C22H22IN3O3
  • MW: 503.33
  • EINECS:
  • MDL Number:MFCD06798331
  • Synonyms:(R)-AM1241;ZUHIXXCLLBMBDW-MRXNPFEDSA-N;(R)-AM1241 Exclusive;(R) AM1241,(R)-AM-1241,(R)AM1241;Methanone, (2-iodo-5-nitrophenyl)[1-[[(2R)-1-methyl-2-piperidinyl]methyl]-1H-indol-3-yl]-
8 prices
Selected condition:
Brand
  • AK Scientific
  • Cayman Chemical
  • TRC
Package
  • 1mg
  • 5mg
  • 10mg
  • 25mg
  • ManufacturerAK Scientific
  • Product number0197DB
  • Product description(R)-(+)-1-((N-Methyl-2-piperidinyl)methyl)-3-(2-iodo-5-nitrobenzoyl)-1H-indole
  • Packaging1mg
  • Price$167
  • Updated2021-12-16
  • Buy
  • ManufacturerAK Scientific
  • Product number0197DB
  • Product description(R)-(+)-1-((N-Methyl-2-piperidinyl)methyl)-3-(2-iodo-5-nitrobenzoyl)-1H-indole
  • Packaging5mg
  • Price$403
  • Updated2021-12-16
  • Buy
  • ManufacturerAK Scientific
  • Product number0197DB
  • Product description(R)-(+)-1-((N-Methyl-2-piperidinyl)methyl)-3-(2-iodo-5-nitrobenzoyl)-1H-indole
  • Packaging25mg
  • Price$1281
  • Updated2021-12-16
  • Buy
  • ManufacturerCayman Chemical
  • Product number10491
  • Product description(R)-AM1241 ≥98%
  • Packaging1mg
  • Price$63
  • Updated2024-03-01
  • Buy
  • ManufacturerCayman Chemical
  • Product number10491
  • Product description(R)-AM1241 ≥98%
  • Packaging5mg
  • Price$275
  • Updated2024-03-01
  • Buy
  • ManufacturerCayman Chemical
  • Product number10491
  • Product description(R)-AM1241 ≥98%
  • Packaging10mg
  • Price$486
  • Updated2024-03-01
  • Buy
  • ManufacturerCayman Chemical
  • Product number10491
  • Product description(R)-AM1241 ≥98%
  • Packaging25mg
  • Price$1062
  • Updated2024-03-01
  • Buy
  • ManufacturerTRC
  • Product numberA729330
  • Product description(R)-AM1241
  • Packaging1mg
  • Price$250
  • Updated2021-12-16
  • Buy
Manufacturer Product number Product description Packaging Price Updated Buy
AK Scientific 0197DB (R)-(+)-1-((N-Methyl-2-piperidinyl)methyl)-3-(2-iodo-5-nitrobenzoyl)-1H-indole 1mg $167 2021-12-16 Buy
AK Scientific 0197DB (R)-(+)-1-((N-Methyl-2-piperidinyl)methyl)-3-(2-iodo-5-nitrobenzoyl)-1H-indole 5mg $403 2021-12-16 Buy
AK Scientific 0197DB (R)-(+)-1-((N-Methyl-2-piperidinyl)methyl)-3-(2-iodo-5-nitrobenzoyl)-1H-indole 25mg $1281 2021-12-16 Buy
Cayman Chemical 10491 (R)-AM1241 ≥98% 1mg $63 2024-03-01 Buy
Cayman Chemical 10491 (R)-AM1241 ≥98% 5mg $275 2024-03-01 Buy
Cayman Chemical 10491 (R)-AM1241 ≥98% 10mg $486 2024-03-01 Buy
Cayman Chemical 10491 (R)-AM1241 ≥98% 25mg $1062 2024-03-01 Buy
TRC A729330 (R)-AM1241 1mg $250 2021-12-16 Buy

Properties

Boiling point :630.7±55.0 °C(Predicted)
Density :1.60±0.1 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :DMF: 25 mg/ml; DMF:PBS(pH7.2) (1:2): 0.3 mg/ml; DMSO: 10 mg/ml; Ethanol: 5 mg/ml
pka :9.73±0.10(Predicted)

Safety Information

Symbol(GHS):
Signal word:
Hazard statements:
Code Hazard statements Hazard class Category Signal word Pictogram P-Codes
Precautionary statements:

Description

(R)-AM1241 avidly binds the peripheral cannabinoid receptor (CB2) (Ki = 15 nM) with over 100-fold selectivity over central cannabinoid receptor (CB1). Like the racemate AM1241 , (R)-AM1241 is an agonist of human CB2, but an inverse agonist of rat and mouse CB2. In rats, (R)-AM1241 produces antinociception to thermal, but not mechanical, pain. The pain-reducing effect of (R)-AM1241 is blocked by the CB2-specific inhibitor SR 144528, but not by either the CB1-selective inhibitor rimonabant or the opioid receptor blocker naloxone.