S1RA
|
- $81 - $2691.1
- Product name: S1RA
- CAS: 878141-96-9
- MF: C20H23N3O2
- MW: 337.42
- EINECS:
- MDL Number:MFCD25976945
- Synonyms:S1RA;4-(2-(5-METHYL-1-(NAPHTHALEN-2-YL)-1H-PYRAZOL-3-YLOXY)ETHYL)MORPHOLINE. HCL;4-[2-[[5-Methyl-1-(2-naphthalenyl)-1H-pyrazol-3-yl]oxy]ethyl]morpholine;4-[2-[[5-Methyl-1-(2-naphthalenyl)-1H-pyrazol-3-yl]oxy]ethyl]morpholine S1RA;S1RA 4-[2-[[5-Methyl-1-(2-naphthalenyl)-1H-pyrazol-3-yl]oxy]ethyl]morpholine;S1RA, >=98%;S1RA, 878141-96-9;4-(2-((5-Methyl-1-(naphthalen-2-yl)-1H-pyrazol-3-yl)oxy)ethyl)morpholine
16 prices
Selected condition：
Brand
- ApexBio Technology
- Biorbyt Ltd
- Cayman Chemical
- Chemenu
- Crysdot
- DC Chemicals
Package
- 500μg
- 1mg
- 5mg
- 10mg
- 25mg
- 50mg
- 100mg
- 250mg
- 1g
- 10mM(in 1mL DMSO)
- 1000mg
- ManufacturerApexBio Technology
- Product numberB1179
- Product descriptionS1RA
- Packaging5mg
- Price$280
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB1179
- Product descriptionS1RA
- Packaging10mM(in 1mL DMSO)
- Price$300
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB1179
- Product descriptionS1RA
- Packaging10mg
- Price$400
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB1179
- Product descriptionS1RA
- Packaging50mg
- Price$1200
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb181123
- Product descriptionS1RA >98%
- Packaging100mg
- Price$765
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb181123
- Product descriptionS1RA >98%
- Packaging250mg
- Price$1504.5
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb181123
- Product descriptionS1RA >98%
- Packaging1000mg
- Price$2691.1
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number16279
- Product descriptionS1RA ≥98%
- Packaging500μg
- Price$81
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number16279
- Product descriptionS1RA ≥98%
- Packaging1mg
- Price$152
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number16279
- Product descriptionS1RA ≥98%
- Packaging5mg
- Price$435
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number16279
- Product descriptionS1RA ≥98%
- Packaging10mg
- Price$711
- Updated2024-03-01
- Buy
- ManufacturerChemenu
- Product numberCM141471
- Product description4-(2-((5-Methyl-1-(naphthalen-2-yl)-1H-pyrazol-3-yl)oxy)ethyl)morpholine 98%
- Packaging100mg
- Price$884
- Updated2021-12-16
- Buy
- ManufacturerCrysdot
- Product numberCD31000448
- Product descriptionS1RA 98+%
- Packaging25mg
- Price$378
- Updated2021-12-16
- Buy
- ManufacturerCrysdot
- Product numberCD31000448
- Product descriptionS1RA 98+%
- Packaging100mg
- Price$945
- Updated2021-12-16
- Buy
- ManufacturerDC Chemicals
- Product numberDC7274
- Product descriptionS1RA >98%
- Packaging100mg
- Price$500
- Updated2021-12-16
- Buy
- ManufacturerDC Chemicals
- Product numberDC7274
- Product descriptionS1RA >98%
- Packaging1g
- Price$1800
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| ApexBio Technology | B1179 | S1RA | 5mg | $280 | 2021-12-16 | Buy |
| ApexBio Technology | B1179 | S1RA | 10mM(in 1mL DMSO) | $300 | 2021-12-16 | Buy |
| ApexBio Technology | B1179 | S1RA | 10mg | $400 | 2021-12-16 | Buy |
| ApexBio Technology | B1179 | S1RA | 50mg | $1200 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb181123 | S1RA >98% | 100mg | $765 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb181123 | S1RA >98% | 250mg | $1504.5 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb181123 | S1RA >98% | 1000mg | $2691.1 | 2021-12-16 | Buy |
| Cayman Chemical | 16279 | S1RA ≥98% | 500μg | $81 | 2024-03-01 | Buy |
| Cayman Chemical | 16279 | S1RA ≥98% | 1mg | $152 | 2024-03-01 | Buy |
| Cayman Chemical | 16279 | S1RA ≥98% | 5mg | $435 | 2024-03-01 | Buy |
| Cayman Chemical | 16279 | S1RA ≥98% | 10mg | $711 | 2024-03-01 | Buy |
| Chemenu | CM141471 | 4-(2-((5-Methyl-1-(naphthalen-2-yl)-1H-pyrazol-3-yl)oxy)ethyl)morpholine 98% | 100mg | $884 | 2021-12-16 | Buy |
| Crysdot | CD31000448 | S1RA 98+% | 25mg | $378 | 2021-12-16 | Buy |
| Crysdot | CD31000448 | S1RA 98+% | 100mg | $945 | 2021-12-16 | Buy |
| DC Chemicals | DC7274 | S1RA >98% | 100mg | $500 | 2021-12-16 | Buy |
| DC Chemicals | DC7274 | S1RA >98% | 1g | $1800 | 2021-12-16 | Buy |
Properties
Boiling point :528.1±50.0 °C(Predicted)
Density :1.21±0.1 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :≥10.35 mg/mL in DMSO; ≥12.23 mg/mL in EtOH; ≥56.1 mg/mL in H2O
form :solid
pka :6.15±0.10(Predicted)
color :Off-white to yellow
Density :1.21±0.1 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :≥10.35 mg/mL in DMSO; ≥12.23 mg/mL in EtOH; ≥56.1 mg/mL in H2O
form :solid
pka :6.15±0.10(Predicted)
color :Off-white to yellow
Safety Information
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| Signal word: | Warning | |||||||||||||||||||||
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Description
The sigma-1 (σ1) receptor is an intracellular, non-opioid receptor that is abundantly expressed in the central nervous system as well as peripherally. S1RA is a potent, selective antagonist of σ1 receptors (Ki = 17 nM) that weakly binds σ2 receptors (Ki = 9,300 nM). It is active in vivo, dose-dependently inhibiting neuropathic pain in several animal models, including formalin-induced nociception and capsaicin-induced mechanical hypersensitivity. S1RA enhances peripheral μ-opioid analgesia without affecting opioid-induced constipation.Suppliers and manufacturers
ATK CHEMICAL COMPANY LIMITED
TargetMol Chemicals Inc.
Zhejiang J&C Biological Technology Co.,Limited
InvivoChem
ShenZhen Trendseen Biological Technology Co.,Ltd.
Wuhan Topule Biopharmaceutical Co., Ltd
LEAPCHEM CO., LTD.
Aladdin Scientific
Amadis Chemical Company Limited
Dalian Meilun Biotech Co., Ltd.