| Company Name: |
TargetMol Chemicals Inc.
|
| Tel: |
15002134094 |
| Email: |
marketing@targetmol.cn |
| Products Intro: |
Product Name:8-CSC
CAS:148589-13-3
Package:100mg/RMB 17500;50mg/RMB 13800;25mg/RMB 10600
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| Company Name: |
CHEMICAL LAND21
|
| Tel: |
82- 2 -783 - 8063 |
| Email: |
sales21@chemicalland21.com |
| Products Intro: |
|
8-(3-chlorostyryl)caffeine manufacturers
- 8-CSC
-
- $2500.00 / 100mg
-
2024-10-28
- CAS:148589-13-3
- Min. Order:
- Purity:
- Supply Ability: 10g
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| | 8-(3-chlorostyryl)caffeine Basic information |
| | 8-(3-chlorostyryl)caffeine Chemical Properties |
| | 8-(3-chlorostyryl)caffeine Usage And Synthesis |
| Uses | 8-(3-Chlorostyryl)caffeine (CSC) is an adenosine antagonist with selective activity at the A2a adenosine receptor. 8-(3-Chlorostyryl)caffeine showed 520-fold selectivity in radioligand binding experiments in rat brain. Antagonism of adenylylase by 8-(3-Chlorostyryl)caffeine shows 22-fold selectivity in rat chromaffin cells When 8-(3-Chlorostyryl)caffeine is co-administered with the A1-selective antagonist CPX, It can also further increase exercise activity. 8-(3-Chlorostyryl)caffeine exhibits good MAO-B inhibitory activity in primate mitochondria. 8-(3-Chlorostyryl)caffeine also has excellent A2A receptor affinity[1]. | | Definition | ChEBI: 8-(3-chlorostyryl)caffeine is caffeine substituted at its 8-position by an (E)-3-chlorostyryl group. It has a role as an adenosine A2A receptor antagonist and an EC 1.4.3.4 (monoamine oxidase) inhibitor. It is a trimethylxanthine and a member of monochlorobenzenes. It is functionally related to a caffeine. | | References | [1] 8-(3-Chlorostyryl)caffeine (CSC) is a selective A2-adenosine antagonist in vitro and in vivo |
| | 8-(3-chlorostyryl)caffeine Preparation Products And Raw materials |
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