| Company Name: |
MedChemexpress LLC
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| Tel: |
021-58955995 |
| Email: |
sales@medchemexpress.cn |
| Products Intro: |
Product Name:CP 316311
CAS:175139-41-0
Purity:>98% Package:5800RMB/1mg
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| Company Name: |
ShangHai Caerulum Pharma Discovery Co., Ltd.
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| Tel: |
18149758185 |
| Email: |
sales-cpd@caerulumpharma.com |
| Products Intro: |
Product Name:3,6-dimethyl-4-pentan-3-yloxy-2-(2,4,6-trimethylphenoxy)pyridine
CAS:175139-41-0
Purity:98% Package:1g;10g;100g
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| Company Name: |
BOC Sciences
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| Tel: |
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| Email: |
info@bocsci.com |
| Products Intro: |
Product Name:CP-316311
CAS:175139-41-0
Purity:98% Remarks:CP-316311, a pyridine derivative, has been found to be a CRF 1 receptor antagonist and was once studied as an antidepressant agent by Pfizer. IC50: 6.8 nM.
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| | CP 316311 Basic information |
| Product Name: | CP 316311 | | Synonyms: | CP 316311;Pyridine, 4-(1-ethylpropoxy)-3,6-dimethyl-2-(2,4,6-trimethylphenoxy)-;3,6-dimethyl-4-pentan-3-yloxy-2-(2,4,6-trimethylphenoxy)pyridine;CP-316 | | CAS: | 175139-41-0 | | MF: | C21H29NO2 | | MW: | 327.46 | | EINECS: | | | Product Categories: | | | Mol File: | 175139-41-0.mol |  |
| | CP 316311 Chemical Properties |
| Melting point | 72.5-74 °C | | Boiling point | 413.9±40.0 °C(Predicted) | | density | 1.007±0.06 g/cm3(Predicted) | | storage temp. | Store at -20°C | | solubility | Soluble in DMSO | | pka | 5.63±0.30(Predicted) |
| | CP 316311 Usage And Synthesis |
| Biological Activity | CP 316311 is a potent and selective CRF1 receptor antagonist with IC50 of 6.8 nM. | | in vitro | CP 316311 fully antagonizes CRF-stimulated adenylate cyclase activity in rat cortex and at human CRF1 receptors endogenously expressed in IMR32 cells with apparent K i values of 7.6 and 8.5 nM, respectively. < /p> | | target | IC50: 6.8 nM (CRF1 receptor) |
| | CP 316311 Preparation Products And Raw materials |
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