Company Name: |
ChemeGen(Shanghai) Biotechnology Co.,Ltd.
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18818260767 |
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sales@chemegen.com |
Products Intro: |
Product Name:XLR11 N-(4-hydroxypentyl) metabolite CAS:1782099-36-8 Purity:98% Package:10 mg;50 mg;100 mg;500 mg;1 g;5 g;10 g
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Company Name: |
Energy Chemical
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Tel: |
021-58432009 400-005-6266 |
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marketing@energy-chemical.com |
Products Intro: |
Product Name:4-Hydroxypentyl XLR11 CAS:1782099-36-8 Purity:NULL Package:100mg;10mg;25mg;50mg Remarks:NULL
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Company Name: |
Shanghai Yifei Biotechnology Co. , Ltd.
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Tel: |
021-65675885 18964387627 |
Email: |
customer_service@efebio.com |
Products Intro: |
Product Name:4-Hydroxypentyl XLR11 CAS:1782099-36-8 Purity:>95% Package:10mg
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Company Name: |
Cayman Chemical Company
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Tel: |
(800) 364-9897 |
Email: |
cayman@caymanchem.com |
Products Intro: |
Product Name:XLR11 N-(4-hydroxypentyl) metabolite (CRM) CAS:1782099-36-8
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| XLR11 N-(4-hydroxypentyl) metabolite (CRM) Basic information |
Product Name: | XLR11 N-(4-hydroxypentyl) metabolite (CRM) | Synonyms: | XLR11 N-(4-hydroxypentyl) metabolite (CRM);[1-(5-fluoro-4-hydroxypentyl)indol-3-yl]-(2,2,3,3-tetramethylcyclopropyl)methanone;XLR11 N-(4-hydroxypentyl) metabolite RM;4-Hydroxypentyl XLR11;XLR-11 4-hydroxypentyl metabolite;XLR11 N-(4-hydroxypentyl) metabolite;Methanone, [1-(5-fluoro-4-hydroxypentyl)-1H-indol-3-yl](2,2,3,3-tetramethylcyclopropyl)- | CAS: | 1782099-36-8 | MF: | C21H28FNO2 | MW: | 345.45 | EINECS: | | Product Categories: | | Mol File: | 1782099-36-8.mol | |
| XLR11 N-(4-hydroxypentyl) metabolite (CRM) Chemical Properties |
Boiling point | 490.0±40.0 °C(Predicted) | density | 1.14±0.1 g/cm3(Predicted) | pka | 13.88±0.20(Predicted) |
| XLR11 N-(4-hydroxypentyl) metabolite (CRM) Usage And Synthesis |
Description | XLR11 is a synthetic cannabinoid (CB) featuring a tetramethylcyclopropyl group, which reportedly confers selectivity for the peripheral CB2 receptor over the central CB1 receptor.1 XLR11 also has an N-(5-fluoropentyl) chain, which increases binding to both CB receptors.2 XLR11 N-(4-hydroxypentyl) metabolite is an expected phase I metabolite of XLR11, based on the known metabolism of similar compounds.3,4 The physiological properties of this compound have not been evaluated. This product is intended for forensic and research applications. | Uses | 4-Hydroxypentyl XLR11 is a metabolite of XLR11 (X746300), an aminoalkylindole compound that is expected to be a cannabinoid (CB) mimetic. | Definition | ChEBI: XLR11 N-(4-hydroxypentyl) metabolite is a member of indoles. | References | 1. Frost, J.M., Dart, M.J., Tietje, K.R., et al. Indol-3-ylcycloalkyl ketones: Effects of N1 substituted indole side chain variations on CB2 cannabinoid receptor activity J. Med. Chem. 53(1),295-315(2010). 2. Makriyannis, A., and Deng, H. Cannabimimetic indole derivatives US7241799B2,(2001). 3. Zhang, Q., Ma, P., Cole, R.B., et al. Identification of in vitro metabolites of JWH-015, an aminoalkylindole agonist for the peripheral cannabinoid receptor (CB2) by HPLC-MS/MS Anal. Bioanal. Chem. 386(5),1345-1355(2006). 4. Wintermeyer, A., M?ller, I., Thevis, M., et al. In vitro phase I metabolism of the synthetic cannabimimetic JWH-018 Anal. Bioanal. Chem. 398(5),2141-2153(2010). |
| XLR11 N-(4-hydroxypentyl) metabolite (CRM) Preparation Products And Raw materials |
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