Company Name: |
3B Pharmachem (Wuhan) International Co.,Ltd.
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Tel: |
821-50328103-801 18930552037 |
Email: |
3bsc@sina.com |
Products Intro: |
Product Name:PSB 11 hydrochloride;(8R)-8-Ethyl-1,4,7,8-tetrahydro-4-5H-iMidazo[2,1-i]purin-5-onehydrochloride CAS:444717-56-0 Purity:99% HPLC Package:1Mg ; 5Mg;10Mg ;100Mg;250Mg ;500Mg ;1g;2.5g ;5g ;10g
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Company Name: |
EMMX Biotechnology LLC
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Tel: |
888-539-0666 |
Email: |
info@emmx.com |
Products Intro: |
Product Name:PSB 11 hydrochloride CAS:444717-56-0 Purity:98% HPLC Package:5mg;10mg;25mg;50mg;100mg;250mg;500mg;1g
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Company Name: |
United States Biological
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Tel: |
1-800-520-3011 |
Email: |
sales@advtechind.com |
Products Intro: |
Product Name:/PSB 11 Hydrochloride
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Company Name: |
United States Biological
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Tel: |
800.520.3011 or 781.639.5092 |
Email: |
chemicals@usbio.net |
Products Intro: |
Product Name:PSB 11 hydrochloride CAS:444717-56-0
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| (8R)-8-ETHYL-1,4,7,8-TETRAHYDRO-4-5H-IMIDAZO[2,1-I]PURIN-5-ONE Basic information |
Product Name: | (8R)-8-ETHYL-1,4,7,8-TETRAHYDRO-4-5H-IMIDAZO[2,1-I]PURIN-5-ONE | Synonyms: | PSB 11 HYDROCHLORIDE;(8R)-8-ETHYL-1,4,7,8-TETRAHYDRO-4-5H-IMIDAZO[2,1-I]PURIN-5-ONE HYDROCHLORIDE;(8R)-8-ETHYL-1,4,7,8-TETRAHYDRO-4-5H-IMIDAZO[2,1-I]PURIN-5-ONE;5H-Imidazo[2,1-i]purin-5-one, 8-ethyl-3,4,7,8-tetrahydro-4-methyl-2-phenyl-, (8R)- | CAS: | 444717-56-0 | MF: | C16H17N5O | MW: | 295.34 | EINECS: | | Product Categories: | | Mol File: | 444717-56-0.mol | |
| (8R)-8-ETHYL-1,4,7,8-TETRAHYDRO-4-5H-IMIDAZO[2,1-I]PURIN-5-ONE Chemical Properties |
storage temp. | Store at +4°C |
| (8R)-8-ETHYL-1,4,7,8-TETRAHYDRO-4-5H-IMIDAZO[2,1-I]PURIN-5-ONE Usage And Synthesis |
Uses | PSB 11 Hydrochloride is a potent and selective antagonist of Adenosine receptor A3-R. | Biological Activity | Potent and selective antagonist for the human adenosine A 3 receptor, with low affinity for the rat A 3 receptor (K i values are 2.3 and > 10000 nM respectively). Displays > 1000-fold selectivity over human A 1 and A 2A receptors (K i values are 4.1 and 3.3 μ M respectively) and > 180-fold selectivity over rat A 1 , rat A 2A and mouse A 2B receptors. Acts as an inverse agonist in the [ 35 S]GTP γ S binding assay in hA 3 -CHO cells (IC 50 = 36 nM). |
| (8R)-8-ETHYL-1,4,7,8-TETRAHYDRO-4-5H-IMIDAZO[2,1-I]PURIN-5-ONE Preparation Products And Raw materials |
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