Company Name: |
3B Pharmachem (Wuhan) International Co.,Ltd.
|
Tel: |
821-50328103-801 18930552037 |
Email: |
3bsc@sina.com |
Products Intro: |
Product Name:Telenzepine dihydrochloride;4,9-Dihydro-3-Methyl-4-[(4-Methyl-1-piperazinyl)acetyl]-10H-thieno[3,4-b][1,5]benzodiazepin-10-onedihydrochloride CAS:147416-96-4 Purity:99% HPLC Package:1Mg ; 5Mg;10Mg ;100Mg;250Mg ;500Mg ;1g;2.5g ;5g ;10g
|
Company Name: |
BOC Sciences
|
Tel: |
1-631-485-4226; 16314854226 |
Email: |
info@bocsci.com |
Products Intro: |
Product Name:Telenzepine dihydrochloride CAS:147416-96-4 Remarks:Telenzepine dihydrochloride is a selective and high affinity muscarinic M1 receptor antagonist (Ki = 0.94 nM). Telenzepine was demonstrated ability to inhibit gastric acid secretion.
|
|
| TELENZEPINE DIHYDROCHLORIDE Basic information |
Product Name: | TELENZEPINE DIHYDROCHLORIDE | Synonyms: | 4,9-DIHYDRO-3-METHYL-4-[(4-METHYL-1-PIPERAZINYL)ACETYL]-10H-THIENO[3,4-B][1,5] BENZODIAZEPIN-10-ONE DIHYDROCHLORIDE;TELENZEPINE DIHYDROCHLORIDE;TELENZEPINE DIHYDROCHLORIDE SELECTIVE M1 MUSCARIN;4,9-Dihydro-3-methyl-4-((4-methyl-1-piperazinyl)acetyl)-(10H)thieno[3,4-b][1,5]benzodiazepin-10-onedihydrochloride;Telenzepine dihydrochloide;Telenzepine hydrate dihydrochloride;4,9-Dihydro-3-methyl-4-((4-methyl-1-piperazinyl)acetyl)-(10H);JTQJFSQQHGPLOX-UHFFFAOYSA-N | CAS: | 147416-96-4 | MF: | C19H22N4O2S | MW: | 370.47 | EINECS: | | Product Categories: | Acetylcholine receptor | Mol File: | 147416-96-4.mol | ![TELENZEPINE DIHYDROCHLORIDE Structure](CAS/GIF/147416-96-4.gif) |
| TELENZEPINE DIHYDROCHLORIDE Chemical Properties |
storage temp. | Store at RT | solubility | H2O: >10 mg/mL | form | solid | color | white | Water Solubility | Soluble to 100 mM in water |
| TELENZEPINE DIHYDROCHLORIDE Usage And Synthesis |
Uses | Telenzepine dihydrochloride is a potent and selective muscarnic receptor antagonist. | Uses | Telenzepine dihydrochloride hydrate was used to study M1 muscarinic receptor-mediated signaling in juvenile rat hippocampus and rat urinary bladder. | Uses | Antiulcerative;M1 muscarinic antagonist | Biological Activity | Selective high affinity muscarinic M 1 receptor antagonist (K i = 0.94 nM). Inhibits gastric acid secretion. | Biochem/physiol Actions | Telenzepine is an analog of pirenzepine and inhibits the secretion of gastric acid. It is an antagonist to M1-receptor and targets the oxyntic gastric glands and the salivary glands. | storage | Desiccate at RT |
| TELENZEPINE DIHYDROCHLORIDE Preparation Products And Raw materials |
|