| Company Name: |
3B Pharmachem (Wuhan) International Co.,Ltd.
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| Tel: |
821-50328103-801 18930552037 |
| Email: |
3bsc@sina.com |
| Products Intro: |
Product Name:L-803,087 trifluoroacetate;N2-[4-(5,7-Difluoro-2-phenyl-1H-indol-3-yl)-1-oxobutyl]-L-arginineMethylestertrifluoroacetate
CAS:217480-26-7
Purity:99% HPLC Package:1Mg ; 5Mg;10Mg ;100Mg;250Mg ;500Mg ;1g;2.5g ;5g ;10g
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| Company Name: |
EMMX Biotechnology LLC
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| Tel: |
888-539-0666 |
| Email: |
info@emmx.com |
| Products Intro: |
Product Name:L-803,087 trifluoroacetate
CAS:217480-26-7
Purity:98% HPLC Package:5mg;10mg;25mg;50mg;100mg;250mg;500mg;1g
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| | L-803,087 TRIFLUOROACETATE Basic information |
| Product Name: | L-803,087 TRIFLUOROACETATE | | Synonyms: | N2-[4-(5,7-DIFLUORO-2-PHENYL-1H-INDOL-3-YL)-1-OXOBUTYL]-L-ARGININE METHYL ESTER TRIFLUOROACETATE;L-803,087 TRIFLUOROACETATE;L-Arginine, N2-[4-(5,7-difluoro-2-phenyl-1H-indol-3-yl)-1-oxobutyl]-, methyl ester;L803087,L 803087 | | CAS: | 217480-26-7 | | MF: | C25H29F2N5O3 | | MW: | 485.53 | | EINECS: | | | Product Categories: | Somatostatin receptor | | Mol File: | 217480-26-7.mol |  |
| | L-803,087 TRIFLUOROACETATE Chemical Properties |
| density | 1.33±0.1 g/cm3(Predicted) | | storage temp. | Store at -20°C | | solubility | Soluble to 100 mM in DMSO and to 100 mM in ethanol | | form | Powder | | pka | 14.54±0.46(Predicted) | | color | White to light yellow |
| | L-803,087 TRIFLUOROACETATE Usage And Synthesis |
| Uses | Somatostatin receptors are often overexpressed in tumours and are potential therapeutic targets. Somatostatin receptor agonists can be used to study signaling pathways related somatostatin receptor. L 803087 is a somatostatin sst4 receptor agonist. | | Biological Activity | Potent and selective somatostatin sst 4 receptor agonist. K i values are 0.7, 199, 4720, 1280 and 3880 nM for cloned human sst 4 , sst 1 , sst 2 , sst 3 and sst 5 receptors respectively. Facilitates AMPA-mediated hippocampal synaptic responses in vitro and increases kainate-induced seizures in mice in vivo . |
| | L-803,087 TRIFLUOROACETATE Preparation Products And Raw materials |
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