中文名:K252b,蛋白激酶抑制剂
英文名:K252b
英文别名:99570-78-2|k-252b|9,12-Epoxy-1H-diindolo[1,2,3-fg:3',2',1'-kl]pyrrolo[3,4-i][1,6]benzodiazocine-10-carboxylicacid, 2,3,9,10,11,12-hexahydro-10-hydroxy-9-methyl-1-oxo-, (9S,10R,12R)-|CHEMBL4750633|(15S,16R,18R)-16-Hydroxy-15-methyl-3-oxo-28-oxa-4,14,19-tri
纯度:≥97%(HPLC)
货号:K139556
包装:100μg
Cas号:99570-78-2
存储温度:-20°C储存
产品介绍:
K252B: an inhibitor of protein kinase A, C, G K-252b is a general, cell permeable protein kinase inhibitor which acts by binding to the ATP binding domain of the kinase. K-252b is a potent inhibitor of CaMKII (Ca2+/calmodulin kinase II), MYLK (myosin light chain kinase, Ki=0.147 μM), PKA (cAMP- dependent protein kinase, Ki=0.09 μM), PKC (protein kinase C, Ki=0.02 μM), and cGKI (cGMP-dependent protein kinase, Ki=0.1 μM).An antibiotic and a strong inhibitor of protein kinase C (PKC)
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关键字: 99570-78-2;k-252b;9,12-Epoxy-1H-diindolo[1,2,3-fg:3',2',1'-kl]pyrrolo[3,4-i][1,6]benzodiazocine-10-carboxylicacid, 2,3,9,10,11,12-hexahydro-10-hydroxy-9-methyl-1-oxo-, (9S,10R,12R)-;CHEMBL4750633
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