中文名:CP-724714
英文名:CP-724714
中文别名:(E)-2-methoxy-N-(3-(4-(3-methyl-4-(6-methylpyridin-3-yloxy)phenylamino)quinazolin-6-yl)allyl)acetamide;2-Methoxy-N-[3-[4-[[3-methyl-4-[(6-methyl-3-pyridinyl)oxy]phenyl]amino]-6-quinazolinyl]-2-propen-1-yl]acetamide
英文别名:(E)-2-methoxy-N-(3-(4-(3-methyl-4-(6-methylpyridin-3-yloxy)phenylamino)quinazolin-6-yl)allyl)acetamide;2-Methoxy-N-[3-[4-[[3-methyl-4-[(6-methyl-3-pyridinyl)oxy]phenyl]amino]-6-quinazolinyl]-2-propen-1-yl]acetamide
纯度:≥99%
货号:C129397
包装:10mg、25mg、50mg
Cas号:537705-08-1
存储温度:-20°C储存
产品介绍:
CP-724714是一种有效的,选择性的HER2/ErbB2抑制剂,IC50为10 nM,比作用于EGFR, InsR, IRG-1R, PDGFR, VEGFR2, Abl, Src, c-Met等选择性高640多倍。Marked selectively against EGFR and potently reduces the EGF-induced autophosphorylation.
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