Салметерол ксинафоат
Салметерол ксинафоат атрибут
| Температура плавления: |
137-138°C |
| температура хранения: |
2-8°C |
| растворимость: |
H2O: мало растворим |
| форма: |
Твердый |
| цвет: |
белый |
| Мерк: |
14,8337 |
| ИнЧИКей: |
XTZNCVSCVHTPAI-UHFFFAOYSA-N |
| Справочник по базе данных CAS: |
94749-08-3(CAS DataBase Reference) |
| FDA UNII: |
6EW8Q962A5 |
| UNSPSC Code: |
41116107 |
| NACRES: |
NA.24 |
Салметерол ксинафоат химические свойства, назначение, производство
Описание
Salmeterol hydroxynaphthoate is a new long-acting β2-selective adrenoceptor agonist
introduced as a bronchodilator for the treatment of reversible airway obstruction in asthma
and chronic bronchitis. It has bronchodilatory activity as intense and four times longerlasting
than equivalent doses of salbutamol. Salmeterol hydroxynaphthoate is reported to
be the first bronchodilator with significant anti-inflammatory activity and hence could
complement prophylactic corticosteroid therapy.
Химические свойства
White to Off-White Solid
Использование
A ?-Adrenergic agonist. Structural analog of albuterol
прикладной
Salmeterol xinafoate is a potent and selective β2-adrenoceptor agonist (EC50 = 5.3 nM) that displays bronchodilator actions. Unlike other β2- adrenoceptor agonists, Salmeterol binds to exo-site domain of β2-AR receptors, producing a slow onset of action and prolonged activation. Clinically used for the treatment of asthma and chronic obstructive pulmonary disease(COPD).
Салметерол ксинафоат препаратная продукция и сырье
сырьё
препарат
Салметерол ксинафоат поставщик
Global( 383)Suppliers
94749-08-3(Салметерол ксинафоат)подобный поиск: