AM 251
|
- $28 - $951
- Product name: AM 251
- CAS: 183232-66-8
- MF: C22H21Cl2IN4O
- MW: 555.24
- EINECS:
- MDL Number:MFCD01861181
- Synonyms:AM 251;1-(2,4-DICHLOROPHENYL)-5-(4-IODOPHENYL)-4-METHYL-N-1-PIPERIDINYL-1 H-PYRAZOLE-3-CARBOXAMIDE;N-(PIPERIDIN-1-YL)-5-(4-IODOPHENYL)-1-(2,4-DICHLOROPHENYL)-4-METHYL-1H-PYRAZOLE-3-CARBOXAMIDE;AM-251 ,99%;AM 251 (pharmaceutical);1H-Pyrazole-3-carboxamide, 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-1-piperidinyl-;1-(2,4-Dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-1-piperidinyl-1H-pyrazole-3-carboxamide AM251;AM251;AM-251
31 prices
Selected condition：
Brand
- ApexBio Technology
- Biorbyt Ltd
- Biosynth Carbosynth
- Cayman Chemical
- Chem-Impex
- ChemScene
- DC Chemicals
- Medical Isotopes, Inc.
- Sigma-Aldrich
- TCI Chemical
- Tocris
- TRC
- Usbiological
Package
- 1
- 1mg
- 50
- 10
- 1unit
- 5mg
- 10mg
- 25mg
- 50mg
- 100mg
- 250mg
- ManufacturerApexBio Technology
- Product numberB1427
- Product descriptionAM 251
- Packaging1unit
- Price$28
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB1427
- Product descriptionAM 251
- Packaging5mg
- Price$40
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB1427
- Product descriptionAM 251
- Packaging10mg
- Price$65
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB1427
- Product descriptionAM 251
- Packaging50mg
- Price$250
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb545947
- Product descriptionAM 251 >98%
- Packaging10mg
- Price$193.8
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb545947
- Product descriptionAM 251 >98%
- Packaging50mg
- Price$538.9
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberBA17338
- Product descriptionAM 251 NEW
- Packaging10mg
- Price$95
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberBA17338
- Product descriptionAM 251 NEW
- Packaging50mg
- Price$332.5
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number71670
- Product descriptionAM 251 ≥98%
- Packaging5mg
- Price$49
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number71670
- Product descriptionAM 251 ≥98%
- Packaging10mg
- Price$92
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number71670
- Product descriptionAM 251 ≥98%
- Packaging50mg
- Price$356
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number71670
- Product descriptionAM 251 ≥98%
- Packaging100mg
- Price$665
- Updated2024-03-01
- Buy
- ManufacturerChem-Impex
- Product number37624
- Product descriptionAM251,97%(HPLC) 97%(HPLC)
- Packaging10MG
- Price$217.28
- Updated2021-12-16
- Buy
- ManufacturerChem-Impex
- Product number37624
- Product descriptionAM251,97%(HPLC) 97%(HPLC)
- Packaging50MG
- Price$733.6
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-3920
- Product descriptionAM 251 98.82%
- Packaging5mg
- Price$50
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-3920
- Product descriptionAM 251 98.82%
- Packaging10mg
- Price$85
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| ApexBio Technology | B1427 | AM 251 | 1unit | $28 | 2021-12-16 | Buy |
| ApexBio Technology | B1427 | AM 251 | 5mg | $40 | 2021-12-16 | Buy |
| ApexBio Technology | B1427 | AM 251 | 10mg | $65 | 2021-12-16 | Buy |
| ApexBio Technology | B1427 | AM 251 | 50mg | $250 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb545947 | AM 251 >98% | 10mg | $193.8 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb545947 | AM 251 >98% | 50mg | $538.9 | 2021-12-16 | Buy |
| Biosynth Carbosynth | BA17338 | AM 251 NEW | 10mg | $95 | 2021-12-16 | Buy |
| Biosynth Carbosynth | BA17338 | AM 251 NEW | 50mg | $332.5 | 2021-12-16 | Buy |
| Cayman Chemical | 71670 | AM 251 ≥98% | 5mg | $49 | 2024-03-01 | Buy |
| Cayman Chemical | 71670 | AM 251 ≥98% | 10mg | $92 | 2024-03-01 | Buy |
| Cayman Chemical | 71670 | AM 251 ≥98% | 50mg | $356 | 2024-03-01 | Buy |
| Cayman Chemical | 71670 | AM 251 ≥98% | 100mg | $665 | 2024-03-01 | Buy |
| Chem-Impex | 37624 | AM251,97%(HPLC) 97%(HPLC) | 10MG | $217.28 | 2021-12-16 | Buy |
| Chem-Impex | 37624 | AM251,97%(HPLC) 97%(HPLC) | 50MG | $733.6 | 2021-12-16 | Buy |
| ChemScene | CS-3920 | AM 251 98.82% | 5mg | $50 | 2021-12-16 | Buy |
| ChemScene | CS-3920 | AM 251 98.82% | 10mg | $85 | 2021-12-16 | Buy |
Properties
Melting point :195-196℃
Density :1.65±0.1 g/cm3(Predicted)
storage temp. :Store at RT
solubility :DMSO: >10 mg/mL, soluble
pka :11.31±0.20(Predicted)
form :solid
color :white
Stability :Stable for 1 year as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.
CAS DataBase Reference :183232-66-8
Density :1.65±0.1 g/cm3(Predicted)
storage temp. :Store at RT
solubility :DMSO: >10 mg/mL, soluble
pka :11.31±0.20(Predicted)
form :solid
color :white
Stability :Stable for 1 year as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.
CAS DataBase Reference :183232-66-8
Safety Information
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Description
SR 141716A is a biarylpyrazole compound which has been considered for many years as the prototypical cannabinoid (CB) receptor antagonist. Some very close structural relatives of SR 141716A were recently prepared and tested for their ability to act as antagonists of the CB1 receptor. AM251 is one of these analogs, wherein the p-chloro group attached to the phenyl substituent at C-5 of the pyrazole ring is replaced with a p-iodo group. The resulting compound exhibits slightly better binding affinity for the CB1 receptor with a Ki value of 7.5 nM compound to SR 141716A, which has a Ki value of 11.5 nM. However AM251 is about two-fold more selective for the CB1 receptor when compared to SR 141716A.More related product prices
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