2-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)ethanamine synthesis

6synthesis methods

Product Name:2-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)ethanamine
CAS Number:138500-90-0
Molecular formula:C14H22BNO2
Molecular Weight:247.141

360792-43-4 Synthesis

tert-butyl 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenethylcarbamate

360792-43-4
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2-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)ethanamine

138500-90-0
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Yield:138500-90-0 91%

Reaction Conditions:

with trifluoroacetic acid in dichloromethane at 20; for 3 h;Cooling with ice;

References:

Liao, Yi;Xu, Liping;Ou, Siyu;Edwards, Holly;Luedtke, Daniel;Ge, Yubin;Qin, Zhihui [ACS Medicinal Chemistry Letters,2018,vol. 9,# 7,p. 635 - 640] Location in patent:supporting information

138500-86-4 Synthesis

4-(Cyanomethyl)benzeneboronic acid pinacol ester

138500-86-4
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$27.00/1g

138500-90-0
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References

68162-47-0
264 suppliers
$13.00/1g

138500-90-0
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References

138500-85-3 Synthesis

4-(Bromomethyl)benzeneboronic acid pinacol ester

138500-85-3
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$8.00/1g

138500-90-0
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References

73918-56-6 Synthesis

73918-56-6
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$20.00/1g

138500-90-0
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References